SCHEMBL29420501

SCHEMBL29420501

COc1ccc(N(N=C(c2ccccc2)c2ccccc2)C(=O)OC(C)(C)C)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.44
CES1 P23141 1/20 0.44
MAPT P10636 5/20 0.43
KMT2A Q03164 5/20 0.43
ALDH1A1 P00352 4/20 0.43
MEN1 O00255 2/20 0.43
GAA P10253 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
KDM4E B2RXH2 1/20 0.42
HPGD P15428 1/20 0.42
MAPK1 P28482 3/20 0.41
TSHR P16473 1/20 0.41
RECQL P46063 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.40
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
CDK5 Q00535 2/20 0.39
CDK5R1 Q15078 2/20 0.39
PKM P14618 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29420512 0.89 KDM4E (0.41) CES2CES1MAPTKMT2AALDH1A1
SCHEMBL29420508 0.89 AAK1 (0.42) KMT2AALDH1A1MEN1SMN1; SMN2HPGD
SCHEMBL29420507 0.87 CES2 (0.39) CES2CES1MAPTKMT2AALDH1A1
SCHEMBL29420485 0.86 AAK1 (0.40) MAPTKMT2AALDH1A1MEN1GAA
SCHEMBL29420493 0.86 MEN1 (0.45) CES2CES1MAPTKMT2AALDH1A1
SCHEMBL29420487 0.86 AAK1 (0.38) MAPTKMT2AALDH1A1MEN1SMN1; SMN2
SCHEMBL29420489 0.86 MEN1 (0.45) CES2CES1MAPTKMT2AALDH1A1
SCHEMBL29420499 0.80 CYP3A4 (0.45) MAPTKMT2AALDH1A1MEN1SMN1; SMN2
SCHEMBL7927967 0.79 CES2 (0.41) CES2CES1MAPTKMT2AALDH1A1
SCHEMBL29420506 0.79 L3MBTL1 (0.47) CES2CES1MAPTKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114195676-B Biarylhydrazine compound and adduct thereof and application of compound in preparation of antitumor drugs 广州药本君安医药科技股份有限公司 2022-08-05 CN disclosed
CN-114195676-A Biarylhydrazine compound and adduct thereof and application of compound in preparation of antitumor drugs 广州药本君安医药科技股份有限公司 2022-03-18 CN disclosed