SCHEMBL29428166

SCHEMBL29428166

COc1ccc(Cn2c(=O)[nH]c3ccc(NC(=O)c4ccccc4OC)cc3c2=O)cc1OC

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.54
TP53 P04637 1/20 0.51
BACE1 P56817 1/20 0.51
KDM4E B2RXH2 3/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
HSD17B10 Q99714 1/20 0.49
CA12 O43570 1/20 0.49
CA9 Q16790 1/20 0.49
KMT2A Q03164 5/20 0.48
ALDH1A1 P00352 3/20 0.48
MEN1 O00255 3/20 0.48
POLB P06746 2/20 0.48
MAPK1 P28482 1/20 0.48
HPGD P15428 1/20 0.48
TOP1 P11387 1/20 0.47
PTGS2 P35354 1/20 0.47
RXFP1 Q9HBX9 1/20 0.47
KCNK3 O14649 1/20 0.47
KCNK9 Q9NPC2 1/20 0.47
HTT P42858 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28699030 1.00 MAPT (0.54) MAPTTP53BACE1KDM4ESMN1; SMN2
SCHEMBL28683077 0.93 MAPT (0.57) MAPTTP53BACE1KDM4ESMN1; SMN2
SCHEMBL29428151 0.85 MAPT (0.54) MAPTTP53BACE1KDM4ESMN1; SMN2
SCHEMBL28685040 0.85 MAPT (0.54) MAPTTP53BACE1KDM4ESMN1; SMN2
SCHEMBL28692022 0.81 SETD7 (0.64) MAPTKMT2AALDH1A1MEN1PTGS2
SCHEMBL29428168 0.81 SETD7 (0.64) MAPTKMT2AALDH1A1MEN1PTGS2
SCHEMBL28692020 0.76 KDM4E (0.61) MAPTTP53BACE1KDM4ESMN1; SMN2
SCHEMBL29428157 0.76 KDM4E (0.61) MAPTTP53BACE1KDM4ESMN1; SMN2
SCHEMBL28694312 0.73 KDM4E (0.56) MAPTTP53BACE1KDM4ESMN1; SMN2
SCHEMBL29428154 0.73 KDM4E (0.56) MAPTTP53BACE1KDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109776434-B 3-benzyl-6-acylamino-2, 4- (1H,3H) -quinazoline diketone derivative and synthesis method and application thereof 中南大学 2022-01-28 CN disclosed