SCHEMBL29428151

SCHEMBL29428151

COc1ccc(Cn2c(=O)[nH]c3ccc(NC(=O)c4cccc(C)c4)cc3c2=O)cc1OC

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.54
TP53 P04637 2/20 0.53
BACE1 P56817 1/20 0.53
KMT2A Q03164 6/20 0.49
MEN1 O00255 3/20 0.49
RXFP1 Q9HBX9 2/20 0.49
ALDH1A1 P00352 3/20 0.48
HPGD P15428 1/20 0.48
KDM4E B2RXH2 4/20 0.47
HSD17B10 Q99714 2/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
ROCK2 O75116 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28685040 1.00 MAPT (0.54) MAPTTP53BACE1KMT2AMEN1
SCHEMBL29428168 0.88 SETD7 (0.64) MAPTKMT2AMEN1ALDH1A1
SCHEMBL28692022 0.88 SETD7 (0.64) MAPTKMT2AMEN1ALDH1A1
SCHEMBL28688249 0.87 ALDH1A1 (0.58) MAPTTP53KMT2AMEN1RXFP1
SCHEMBL29428166 0.85 MAPT (0.54) MAPTTP53BACE1KMT2AMEN1
SCHEMBL28699030 0.85 MAPT (0.54) MAPTTP53BACE1KMT2AMEN1
SCHEMBL14363190 0.78 KCNK3 (0.68) MAPTTP53KMT2AMEN1RXFP1
SCHEMBL28683077 0.77 MAPT (0.57) MAPTTP53BACE1KMT2AMEN1
SCHEMBL29428157 0.74 KDM4E (0.61) MAPTTP53BACE1KMT2AMEN1
SCHEMBL28692020 0.74 KDM4E (0.61) MAPTTP53BACE1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109776434-B 3-benzyl-6-acylamino-2, 4- (1H,3H) -quinazoline diketone derivative and synthesis method and application thereof 中南大学 2022-01-28 CN disclosed