SCHEMBL28683077

SCHEMBL28683077

COc1ccccc1C(=O)Nc1ccc2[nH]c(=O)n(Cc3ccccc3)c(=O)c2c1

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.57
CA12 O43570 2/20 0.55
CA9 Q16790 2/20 0.55
TSHR P16473 1/20 0.52
MAPK1 P28482 1/20 0.52
TP53 P04637 1/20 0.52
BACE1 P56817 1/20 0.52
ALDH1A1 P00352 6/20 0.51
KDM4E B2RXH2 5/20 0.51
KMT2A Q03164 4/20 0.51
MEN1 O00255 3/20 0.50
KCNK3 O14649 2/20 0.50
KCNK9 Q9NPC2 2/20 0.50
POLB P06746 1/20 0.50
RXFP1 Q9HBX9 1/20 0.50
BRPF1 P55201 1/20 0.49
HPGD P15428 2/20 0.49
CASP3 P42574 2/20 0.48
SMN1; SMN2 Q16637 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29428166 0.93 MAPT (0.54) MAPTCA12CA9MAPK1TP53
SCHEMBL28699030 0.93 MAPT (0.54) MAPTCA12CA9MAPK1TP53
SCHEMBL28688249 0.79 ALDH1A1 (0.58) MAPTCA12CA9TP53ALDH1A1
SCHEMBL29428151 0.77 MAPT (0.54) MAPTTP53BACE1ALDH1A1KDM4E
SCHEMBL28685040 0.77 MAPT (0.54) MAPTTP53BACE1ALDH1A1KDM4E
SCHEMBL6243745 0.76 MAPT (0.60) MAPTTSHRMAPK1TP53BACE1
SCHEMBL28683072 0.74 MEN1 (0.58) MAPTALDH1A1KMT2AMEN1POLB
SCHEMBL29428168 0.74 SETD7 (0.64) MAPTALDH1A1KMT2AMEN1
SCHEMBL28692022 0.74 SETD7 (0.64) MAPTALDH1A1KMT2AMEN1
SCHEMBL10085009 0.73 KDM4E (0.68) MAPTALDH1A1KDM4EKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109776434-B 3-benzyl-6-acylamino-2, 4- (1H,3H) -quinazoline diketone derivative and synthesis method and application thereof 中南大学 2022-01-28 CN disclosed