SCHEMBL29433296

SCHEMBL29433296

CON(C)C(=O)C(F)(F)c1cccc(N)c1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.46
MAPK1 P28482 1/20 0.46
MLYCD O95822 1/20 0.38
PTGS1 P23219 4/20 0.38
ALDH1A1 P00352 3/20 0.37
NPSR1 Q6W5P4 1/20 0.36
TP53 P04637 1/20 0.35
CYP3A4 P08684 1/20 0.35
CLK1 P49759 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
CFTR P13569 1/20 0.33
KDM1A O60341 1/20 0.33
HSD11B1 P28845 1/20 0.33
MAOB P27338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22670274 1.00 TSHR (0.46) TSHRMAPK1MLYCDPTGS1ALDH1A1
SCHEMBL25006865 0.82 RIPK1 (0.41) MLYCDALDH1A1CYP3A4CLK1HSD11B1
SCHEMBL30222838 0.82 RIPK1 (0.41) MLYCDALDH1A1CYP3A4CLK1HSD11B1
SCHEMBL25007307 0.81 PTPN5 (0.48)
SCHEMBL30222787 0.81 PTPN5 (0.48)
SCHEMBL22165138 0.78 TSHR (0.52) TSHRMAPK1PTGS1ALDH1A1NPSR1
SCHEMBL22658398 0.78 TP53 (0.50) ALDH1A1NPSR1TP53SMN1; SMN2
SCHEMBL22670292 0.74 RXFP1 (0.52) ALDH1A1NPSR1TP53SMN1; SMN2
SCHEMBL15272073 0.74 TSHR (0.59) TSHRMAPK1PTGS1ALDH1A1CYP3A4
SCHEMBL30707942 0.74 TSHR (0.59) TSHRMAPK1PTGS1ALDH1A1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3983386-A1 ACSS2 INHIBITORS AND METHODS OF USE THEREOF Metabomed Ltd (IL) 2022-04-20 EP disclosed
CN-114008025-A ACSS2 inhibitors and methods of use thereof 美特波米德有限公司 2022-02-01 CN disclosed