SCHEMBL29435582

SCHEMBL29435582

CSC(=N)Nc1ncc(C(F)(F)F)cc1N(C)C(=O)OC(C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.37
MEN1 O00255 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
ALDH1A1 P00352 5/20 0.36
KDM4E B2RXH2 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
MAPK1 P28482 1/20 0.34
LIPE Q05469 4/20 0.34
HPGD P15428 1/20 0.33
ABL1 P00519 1/20 0.33
CACNA1G O43497 1/20 0.33
CACNA1B Q00975 1/20 0.33
CACNA1C Q13936 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22583033 1.00 KMT2A (0.37) KMT2AMEN1SMN1; SMN2ALDH1A1KDM4E
SCHEMBL22583237 0.85 SMN1; SMN2 (0.40) KMT2AMEN1SMN1; SMN2ALDH1A1KDM4E
SCHEMBL22583484 0.83 ALDH1A1 (0.39) KMT2AMEN1SMN1; SMN2ALDH1A1KDM4E
SCHEMBL29601868 0.83 ALDH1A1 (0.39) KMT2AMEN1SMN1; SMN2ALDH1A1KDM4E
SCHEMBL22583431 0.81 BACE1 (0.34) KMT2AMEN1LIPEABL1CACNA1G
SCHEMBL29435649 0.81 BACE1 (0.34) KMT2AMEN1LIPEABL1CACNA1G
SCHEMBL29435524 0.76 ALDH1A1 (0.41) KMT2AMEN1SMN1; SMN2ALDH1A1KDM4E
SCHEMBL22583372 0.76 ALDH1A1 (0.41) KMT2AMEN1SMN1; SMN2ALDH1A1KDM4E
SCHEMBL22583020 0.76 ALDH1A1 (0.38) KMT2AMEN1ALDH1A1KDM4EMAPK1
SCHEMBL29435611 0.76 ALDH1A1 (0.43) KMT2AMEN1SMN1; SMN2ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250276967-A1 HETEROCYCLIC COMPOUNDS AND THEIR USE FOR TREATMENT OF HELMINTHIC INFECTIONS AND DISEASES SIGNAL PHARMACEUTICALS, LLC 2025-09-04 US disclosed
US-12338235-B2 Heterocyclic compounds and their use for treatment of helminthic infections and diseases CELGENE CORPORATION (US) 2025-06-24 US disclosed
US-11505548-B2 Heterocyclic compounds and their use for treatment of helminthic infections and diseases CELGENE CORPORATION (US) 2022-11-22 US disclosed
EP-3959207-A1 HETEROCYCLIC COMPOUNDS AND THEIR USE FOR TREATMENT OF HELMINTHIC INFECTIONS AND DISEASES Celgene Corporation (US) 2022-03-02 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250276967-A1 HETEROCYCLIC COMPOUNDS AND THEIR USE FOR TREATMENT OF HELMINTHIC INFECTIONS AND DISEASES CYP8B1, HAX1, HRH4 KMT2A 3502/4885MEN1 2158/4885SMN1; SMN2 668/4885
US-11505548-B2 Heterocyclic compounds and their use for treatment of helminthic infections and diseases CYP8B1, HAX1, HRH4 KMT2A 3502/4885MEN1 2158/4885SMN1; SMN2 668/4885
US-12338235-B2 Heterocyclic compounds and their use for treatment of helminthic infections and diseases CYP8B1, HAX1, HRH4 KMT2A 3502/4885MEN1 2158/4885SMN1; SMN2 668/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.