SCHEMBL29439864

SCHEMBL29439864

Clc1ncnc2c1CN(c1cccc(I)c1)CC2

nearest known ligand 0.37

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 10/20 0.37
P2RX2 Q9UBL9 4/20 0.37
PIK3CD O00329 3/20 0.37
TRPV1 Q8NER1 1/20 0.33
PIK3CA P42336 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22715552 1.00 P2RX3 (0.37) P2RX3P2RX2PIK3CDTRPV1PIK3CA
SCHEMBL22715950 0.85 PIK3CD (0.37) P2RX3P2RX2PIK3CDPIK3CA
SCHEMBL29439836 0.85 PIK3CD (0.37) P2RX3P2RX2PIK3CDPIK3CA
SCHEMBL22715558 0.85 PIK3CD (0.37) P2RX3P2RX2PIK3CDPIK3CA
SCHEMBL29439669 0.85 PIK3CD (0.37) P2RX3P2RX2PIK3CDPIK3CA
SCHEMBL23870044 0.78 IP6K1 (0.39) PIK3CD
SCHEMBL29439678 0.78 IP6K1 (0.39) PIK3CD
SCHEMBL2849692 0.72 GRIN2D (0.52) P2RX3PIK3CDPIK3CA
SCHEMBL8088154 0.72 KDM4E (0.47) P2RX3P2RX2
SCHEMBL2849660 0.71 TRPV1 (0.53) P2RX3TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118908957-A Small molecule inhibitors of NF- κB induced kinase 詹森药业有限公司 2024-11-08 CN disclosed
CN-114222737-B Small molecule inhibitors of NF- κB induced kinase 詹森药业有限公司 2024-07-26 CN disclosed
EP-3976597-A1 SMALL MOLECULE INHIBITORS OF NF-KB INDUCING KINASE Janssen Pharmaceutica NV (BE) 2022-04-06 EP disclosed