SCHEMBL29443012

SCHEMBL29443012

O=C1N(c2ccc(Br)cc2)CCC12Cc1ccc(F)cc1C2

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HDAC11 Q96DB2 4/20 0.38
MAPT P10636 3/20 0.37
DOCK5 Q9H7D0 1/20 0.36
METAP2 P50579 3/20 0.35
MEN1 O00255 1/20 0.35
MAPK1 P28482 1/20 0.35
KMT2A Q03164 1/20 0.35
FPR2 P25090 1/20 0.34
OTUD7B Q6GQQ9 1/20 0.34
CXCR3 P49682 1/20 0.34
EBP Q15125 1/20 0.33
LIPE Q05469 1/20 0.33
AVPR1A P37288 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21490366 1.00 HDAC11 (0.38) HDAC11MAPTDOCK5METAP2MEN1
SCHEMBL29443074 0.84 HDAC11 (0.42) HDAC11MAPTMEN1KMT2ALIPE
SCHEMBL21490337 0.84 HDAC11 (0.42) HDAC11MAPTMEN1KMT2ALIPE
SCHEMBL21490362 0.82 ROCK2 (0.44) OTUD7BLIPEAVPR1A
SCHEMBL29443020 0.82 ROCK2 (0.44) OTUD7BLIPEAVPR1A
SCHEMBL21084133 0.79 HDAC11 (0.47) HDAC11METAP2
SCHEMBL21084147 0.79 HDAC11 (0.47) HDAC11METAP2
SCHEMBL22355673 0.79 ITGB3 (0.38) HDAC11DOCK5METAP2LIPE
SCHEMBL21490367 0.79 ROCK2 (0.49)
SCHEMBL29442925 0.79 ROCK2 (0.49)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689639-B Spirolactams as ROCK inhibitors 百时美施贵宝公司 2022-02-18 CN disclosed