SCHEMBL22355673

SCHEMBL22355673

N=C/C(=C\N)c1ccc(N2CCC3(Cc4ccc(F)cc4C3)C2=O)cc1

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 13/20 0.38
ITGA2B P08514 13/20 0.38
METAP2 P50579 2/20 0.35
HDAC11 Q96DB2 2/20 0.33
HTR2C P28335 1/20 0.32
HRH1 P35367 1/20 0.32
LIPE Q05469 1/20 0.32
DOCK5 Q9H7D0 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22355757 0.88 ITGB3 (0.41) ITGB3ITGA2BHDAC11
SCHEMBL22355671 0.86 ITGB3 (0.37) ITGB3ITGA2BLIPE
SCHEMBL22355676 0.81 ROCK2 (0.43) METAP2
SCHEMBL29443012 0.79 HDAC11 (0.38) METAP2HDAC11LIPEDOCK5
SCHEMBL21490366 0.79 HDAC11 (0.38) METAP2HDAC11LIPEDOCK5
SCHEMBL24742882 0.78 ITGB3 (0.44) ITGB3ITGA2BLIPE
SCHEMBL24742787 0.77 HSD11B1 (0.42) ITGB3ITGA2B
SCHEMBL24743240 0.76 ITGB3 (0.40) ITGB3ITGA2BLIPE
SCHEMBL22355680 0.76 BACE1 (0.33) HDAC11
SCHEMBL21084147 0.75 HDAC11 (0.47) ITGB3ITGA2BMETAP2HDAC11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3481817-B1 SPIROLACTAMS AS INHIBITORS OF ROCK BRISTOL MYERS SQUIBB CO (US) 2020-08-19 EP disclosed