SCHEMBL29444510

SCHEMBL29444510

NN=C1C(=O)Nc2c(F)ccc(Br)c21

nearest known ligand 0.34

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 1/20 0.34
ABCC8 Q09428 1/20 0.34
KCNJ11 Q14654 1/20 0.34
KCNJ8 Q15842 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19210975 1.00 ABCC9 (0.34) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL19210856 1.00 ABCC9 (0.34) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL29444533 0.78 CES1 (0.41) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL19210912 0.78 CES1 (0.41) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL32662403 0.74 CA1 (0.32)
SCHEMBL5988227 0.69 CES1 (0.44)
SCHEMBL5739112 0.68 CES1 (0.50)
SCHEMBL5739017 0.68 CA1 (0.41)
SCHEMBL24399769 0.67 TGM2 (0.43) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL5740135 0.66 CES1 (0.58)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108884096-B Spiroindolinones as DDR1 inhibitors 豪夫迈·罗氏有限公司 2022-03-22 CN disclosed