SCHEMBL29444533

SCHEMBL29444533

O=C1Nc2c(F)ccc(Br)c2C1=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 12/20 0.41
TGM2 P21980 2/20 0.39
ALDH1A1 P00352 2/20 0.37
ALDH2 P05091 1/20 0.37
ALDH3A1 P30838 1/20 0.37
DNMT1 P26358 1/20 0.35
ABCC9 O60706 2/20 0.35
ABCC8 Q09428 2/20 0.35
KCNJ11 Q14654 2/20 0.35
KCNJ8 Q15842 2/20 0.35
DAO P14920 2/20 0.32
BCHE P06276 2/20 0.32
NSD2 O96028 1/20 0.32
MEN1 O00255 1/20 0.31
POLB P06746 1/20 0.31
MAPT P10636 1/20 0.31
HTT P42858 1/20 0.31
KMT2A Q03164 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
CDK2 P24941 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19210912 1.00 CES1 (0.41) CES1TGM2ALDH1A1ALDH2ALDH3A1
SCHEMBL24399769 0.85 TGM2 (0.43) CES1TGM2ALDH1A1ALDH2ALDH3A1
SCHEMBL17265675 0.84 CES1 (0.47) CES1TGM2ALDH1A1ALDH2ALDH3A1
SCHEMBL331905 0.84 TGM2 (0.48) CES1TGM2DNMT1DAOBCHE
SCHEMBL19210975 0.78 ABCC9 (0.34) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL19210856 0.78 ABCC9 (0.34) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL29444510 0.78 ABCC9 (0.34) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL31528208 0.77 CES1 (0.71) CES1TGM2ALDH1A1ALDH2ALDH3A1
SCHEMBL20505489 0.77 CES1 (0.71) CES1TGM2DNMT1DAOBCHE
SCHEMBL31728064 0.77 CES1 (0.41) CES1TGM2ALDH1A1ALDH2ALDH3A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113801053-B Method for preparing 7-fluoro-2-oxoindoline-4-carboxylic acid 上海皓鸿生物医药科技有限公司 2023-09-08 CN claimed
CN-113801053-B Method for preparing 7-fluoro-2-oxoindoline-4-carboxylic acid 上海皓鸿生物医药科技有限公司 2023-09-08 CN disclosed
CN-113801053-B Method for preparing 7-fluoro-2-oxoindoline-4-carboxylic acid 上海皓鸿生物医药科技有限公司 2023-09-08 CN disclosed
CN-108884096-B Spiroindolinones as DDR1 inhibitors 豪夫迈·罗氏有限公司 2022-03-22 CN disclosed