Voriconazole

Voriconazole

SCHEMBL29449336

C[C@@H](c1ncncc1F)[C@](O)(Cn1cncn1)c1ccc(F)cc1F

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ERG11

The experimentally established mechanism targets of Voriconazole. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 17/20 1.00
CYP2C9 P11712 11/20 1.00
CYP2C19 P33261 11/20 1.00
LMNA P02545 2/20 1.00
CYP2B6 P20813 1/20 1.00
CYP3A5 P20815 1/20 1.00
CYP3A7 P24462 1/20 1.00
MAPK1 P28482 1/20 1.00
CYP3A43 Q9HB55 1/20 1.00
CYP46A1 Q9Y6A2 1/20 1.00
HSP90AA1 P07900 1/20 0.58
CYP19A1 P11511 1/20 0.58
CYP11B1 P15538 1/20 0.58
CYP11B2 P19099 1/20 0.58
ADRA1A P35348 1/20 0.58
CYP51A1 Q16850 1/20 0.58
CYP1A2 P05177 6/20 0.56
CYP2D6 P10635 6/20 0.56
KCNH2 Q12809 3/20 0.56
ABCG2 Q9UNQ0 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Voriconazole SCHEMBL29449338 1.00 CYP3A4 (1.00) CYP3A4CYP2C9CYP2C19LMNACYP2B6
Voriconazole SCHEMBL28720611 1.00 CYP3A4 (1.00) CYP3A4CYP2C9CYP2C19LMNACYP2B6
Voriconazole SCHEMBL824156 1.00 CYP3A4 (1.00) CYP3A4CYP2C9CYP2C19LMNACYP2B6
Voriconazole SCHEMBL1554444 1.00 CYP3A4 (1.00) CYP3A4CYP2C9CYP2C19LMNACYP2B6
Voriconazole SCHEMBL29378592 1.00 CYP3A4 (1.00) CYP3A4CYP2C9CYP2C19LMNACYP2B6
Voriconazole SCHEMBL29449335 1.00 CYP3A4 (1.00) CYP3A4CYP2C9CYP2C19LMNACYP2B6
Voriconazole SCHEMBL371715 1.00 CYP3A4 (1.00) CYP3A4CYP2C9CYP2C19LMNACYP2B6
Voriconazole SCHEMBL3949267 1.00 CYP3A4 (1.00) CYP3A4CYP2C9CYP2C19LMNACYP2B6
Voriconazole SCHEMBL4709722 1.00 CYP3A4 (1.00) CYP3A4CYP2C9CYP2C19LMNACYP2B6
Voriconazole SCHEMBL3713297 1.00 CYP3A4 (1.00) CYP3A4CYP2C9CYP2C19LMNACYP2B6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 36 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025215232-A1 A COMPOSITION COMPRISING A SAPONIN AND/OR AN ANTHELMINTIC AND/OR A MITOCHONDRIAL UNCOUPLER FOR THE TREATMENT OF LIVER DISEASE RAINCASTLE BIO. LIMITED (GB) 2025-10-16 WO claimed
CN-119510476-A Voriconazole structure identification method based on multidimensional nuclear magnetic resonance 武汉商学院 2025-02-25 CN claimed
EP-4019509-A1 METHOD FOR PREPARING VORICONAZOLE L-CAMPHORSULPHONATE Zhejiang Huahai Pharmaceutical Co., Ltd (CN) 2022-06-29 EP claimed
EP-4633677-A1 VIROPORINS BLOCKERS/INHIBITORS AS ANTI-INFLUENZA AGENTS Yissum Research Development Company of the Hebrew University of Jerusalem Ltd. (IL) 2025-10-22 EP disclosed
CN-119868580-A Cyclodextrin inclusion compound and preparation method thereof 江苏东科康德药业有限公司 2025-04-25 CN disclosed
CN-119823105-A Preparation method of racemic voriconazole 苏州第四制药厂有限公司 2025-04-15 CN disclosed
CN-119564599-A Preparation process of voriconazole intermediate liquid medicine for injection 湖南赛隆药业(长沙)有限公司 2025-03-07 CN disclosed
CN-119555826-A Method for detecting 4- (1, 1-dibromoethyl) -6-chloro-5-fluoropyrimidine in voriconazole 珠海润都制药股份有限公司 2025-03-04 CN disclosed
CN-119510476-A Voriconazole structure identification method based on multidimensional nuclear magnetic resonance 武汉商学院 2025-02-25 CN disclosed
CN-119499192-A Preparation method of voriconazole for injection 湖南赛隆药业(长沙)有限公司 2025-02-25 CN disclosed
CN-119306703-A Synthesis method of voriconazole 湖北午时医药研究院有限公司 2025-01-14 CN disclosed
CN-106432198-B Method for preparing voriconazole split intermediate 浙江华海药业股份有限公司 2022-10-21 CN disclosed
CN-114965912-A Voriconazole structure detection method based on spectrum characteristics 丁力 2022-08-30 CN disclosed
US-20220213073-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF FUNGAL INFECTIONS CELLIX BIO PRIVATE LIMITED (IN) 2022-07-07 US disclosed
EP-4019509-A1 METHOD FOR PREPARING VORICONAZOLE L-CAMPHORSULPHONATE Zhejiang Huahai Pharmaceutical Co., Ltd (CN) 2022-06-29 EP disclosed
CN-112898273-B Synthetic method and application of voriconazole 海南锦瑞制药有限公司 2022-05-31 CN disclosed
US-11312707-B2 Compositions and methods for the treatment of fungal infections CELLIX BIO PRIVATE LIMITED (IN) 2022-04-26 US disclosed
CN-114344245-A Voriconazole external preparation and preparation method thereof 浙江普利药业有限公司 2022-04-15 CN disclosed
CN-114191387-A Preparation method of voriconazole oral liquid 苏州海景医药科技有限公司 2022-03-18 CN disclosed
EP-3511326-B1 METHOD FOR PREPARING VORICONAZOLE L-CAMPHORSULPHONATE AND VORICONAZOLE ZHEJIANG HUAHAI PHARM CO LTD (CN) 2022-03-09 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11312707-B2 Compositions and methods for the treatment of fungal infections SI, CYP3A7, ERG28 CYP3A4 4/4885CYP2C9 31/4885CYP2C19 40/4885
US-20220213073-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF FUNGAL INFECTIONS SI, CYP3A7, ERG28 CYP3A4 4/4885CYP2C9 31/4885CYP2C19 40/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.