SCHEMBL29450481

SCHEMBL29450481

COC(=O)c1ccc(Cl)nc1Cl

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TUBB4A P04350 1/20 0.54
TUBB P07437 1/20 0.54
TUBA3C P0DPH7 1/20 0.54
TUBA1B P68363 1/20 0.54
TUBA4A P68366 1/20 0.54
TUBB4B P68371 1/20 0.54
TUBB3 Q13509 1/20 0.54
TUBB2A Q13885 1/20 0.54
TUBB8 Q3ZCM7 1/20 0.54
TUBA3E Q6PEY2 1/20 0.54
TUBA1A Q71U36 1/20 0.54
TUBA1C Q9BQE3 1/20 0.54
TUBB6 Q9BUF5 1/20 0.54
TUBB2B Q9BVA1 1/20 0.54
TUBB1 Q9H4B7 1/20 0.54
KDM4E B2RXH2 4/20 0.49
SMN1; SMN2 Q16637 3/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
NPC1 O15118 2/20 0.47
MAPT P10636 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL424747 1.00 TUBB4A (0.54) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL2032206 0.85 ABL1 (0.53) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL29416399 0.83 TUBB4A (0.52) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL1246770 0.83 SMN1; SMN2 (0.62) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL30798551 0.83 SMN1; SMN2 (0.62) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL24818230 0.83 LMNA (0.48) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL1615811 0.83 NPC1 (0.46) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL3051920 0.83 TUBB4A (0.52) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL334079 0.83 EGFR (0.50) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL29453741 0.83 EGFR (0.50) TUBB4ATUBBTUBA3CTUBA1BTUBA4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122036605-A Antagonists of GPR39 proteins 俄勒冈健康科学大学 2026-05-15 CN disclosed
CN-119630670-A Modulators of TNFalpha activity and uses thereof 瑞雷拉公司 2025-03-14 CN disclosed
EP-4463456-A1 THIAZOLOPYRIDYL AMIDE DERIVATIVES AS DNA POLYMERASE THETA INHIBITORS BeiGene, Ltd. (KY) 2024-11-20 EP disclosed
CN-116554151-B Kinesin KIF18A inhibitor and application thereof 上海湃隆生物科技有限公司 2024-09-20 CN disclosed
CN-118510778-A Thiazolopyridylamide derivatives as inhibitors of DNA polymerase θ 百济神州有限公司 2024-08-16 CN disclosed
CN-116554151-A Kinesin KIF18A inhibitor and application thereof 上海湃隆生物科技有限公司 2023-08-08 CN disclosed
WO-2023134708-A1 THIAZOLOPYRIDYL AMIDE DERIVATIVES AS DNA POLYMERASE THETA INHIBITORS BEIGENE , LTD. (KY) 2023-07-20 WO disclosed
CN-115996908-A Antagonists of GPR39 proteins 俄勒冈健康科学大学 2023-04-21 CN disclosed
CN-114391015-A Benzo [ b ] [1,8] naphthyridineacetic acid derivatives and methods of use 斯汀塞拉股份有限公司 2022-04-22 CN disclosed
EP-3969452-A1 BENZO[B][1,8]NAPHTHYRIDINE ACETIC ACID DERIVATIVES AND METHODS OF USE Stingthera, Inc. (US) 2022-03-23 EP disclosed