SCHEMBL29463590

SCHEMBL29463590

COC(=O)c1cc(=O)c2ccc(OS(=O)(=O)C(F)(F)F)cc2o1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.69
ALDH1A1 P00352 4/20 0.56
HSD11B1 P28845 1/20 0.49
EPHX2 P34913 1/20 0.47
SLC2A1 P11166 1/20 0.46
AKR1B1 P15121 4/20 0.45
MAPT P10636 3/20 0.44
GAA P10253 1/20 0.44
LMNA P02545 2/20 0.44
KMT2A Q03164 2/20 0.44
NPSR1 Q6W5P4 1/20 0.44
TSHR P16473 1/20 0.44
THRB P10828 1/20 0.44
AR P10275 1/20 0.43
ACHE P22303 1/20 0.42
MEN1 O00255 1/20 0.42
TP53 P04637 1/20 0.42
CYP3A4 P08684 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
STS P08842 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2812506 0.87 AKR1B1 (0.62) KDM4EALDH1A1HSD11B1EPHX2SLC2A1
SCHEMBL8107875 0.82 KDM4E (1.00) KDM4EALDH1A1EPHX2SLC2A1AKR1B1
SCHEMBL2810641 0.81 PIM1 (0.56) KDM4EALDH1A1HSD11B1MAPTLMNA
SCHEMBL1500205 0.80 EPHX2 (0.54) KDM4EALDH1A1HSD11B1EPHX2MAPT
SCHEMBL1500319 0.80 EPHX2 (0.50) KDM4EALDH1A1HSD11B1EPHX2GAA
SCHEMBL2083018 0.80 SMN1; SMN2 (0.49) KDM4EALDH1A1HSD11B1MAPTGAA
SCHEMBL8107014 0.78 KDM4E (0.76) KDM4EALDH1A1SLC2A1AKR1B1MAPT
SCHEMBL8107902 0.76 KDM4E (0.72) KDM4EALDH1A1SLC2A1AKR1B1MAPT
SCHEMBL8119217 0.75 AKR1B1 (0.74) KDM4EALDH1A1AKR1B1GAAKMT2A
SCHEMBL4254491 0.75 KDM4E (0.72) KDM4EALDH1A1SLC2A1AKR1B1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022036040-A1 SYNTHESIS OF SMALL MOLECULES INSPIRED BY PHOMOXANTHONE A WORCESTER POLYTECHNIC INSTITUTE (US) 2022-02-17 WO disclosed