SCHEMBL2947210

SCHEMBL2947210

CCc1ccccc1-c1ccc(C#N)c(F)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 14/20 0.51
CYP11B2 P19099 14/20 0.51
ALOX5AP P20292 1/20 0.49
FEN1 P39748 1/20 0.49
TUBB4A P04350 1/20 0.48
TUBB P07437 1/20 0.48
TUBA3C P0DPH7 1/20 0.48
STAT3 P40763 1/20 0.48
TUBA1B P68363 1/20 0.48
TUBA4A P68366 1/20 0.48
TUBB4B P68371 1/20 0.48
TUBB3 Q13509 1/20 0.48
TUBB2A Q13885 1/20 0.48
TUBB8 Q3ZCM7 1/20 0.48
TUBA3E Q6PEY2 1/20 0.48
TUBA1A Q71U36 1/20 0.48
TUBA1C Q9BQE3 1/20 0.48
TUBB6 Q9BUF5 1/20 0.48
TUBB2B Q9BVA1 1/20 0.48
TUBB1 Q9H4B7 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23347204 0.80 ALOX5AP (0.56) ALOX5APFEN1STAT3TRPA1
SCHEMBL3304437 0.80 CYP11B1 (0.72) CYP11B1CYP11B2TUBB4ATUBBTUBA3C
SCHEMBL14555723 0.78 CYP11B1 (0.68) CYP11B1CYP11B2ALOX5APFEN1TUBB4A
SCHEMBL8678897 0.76 SYK (0.43) CYP11B1CYP11B2TUBB4ATUBBTUBA3C
SCHEMBL24989659 0.76 CYP11B1 (0.48) CYP11B1CYP11B2KCNJ1
SCHEMBL9755559 0.75 TSHR (0.49) CYP11B1CYP11B2TUBB4ATUBBTUBA3C
SCHEMBL9287992 0.75 ALOX5AP (0.50) ALOX5APFEN1TRPA1
SCHEMBL2948017 0.75 ALOX5AP (0.54) ALOX5APFEN1TRPA1
SCHEMBL21675486 0.75 ALOX5AP (0.42) ALOX5APFEN1TRPA1
SCHEMBL19187744 0.74 CYP11B1 (0.54) CYP11B1CYP11B2KCNJ1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2396301-A2 SMALL MOLECULE BRADYKININ B1 RECEPTOR ANTAGONISTS Jerini AG (DE) 2011-12-21 EP disclosed
WO-2010091876-A2 SMALL MOLECULE BRADYKININ B1 RECEPTOR ANTAGONISTS JERINI AG (DE) 2010-08-19 WO disclosed