SCHEMBL29478786

SCHEMBL29478786

O=C(O)c1cc(C(F)(F)F)nn1Cc1cccnc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SORT1 Q99523 7/20 0.57
GRN P28799 6/20 0.57
MARS1 P56192 2/20 0.53
KLKB1 P03952 1/20 0.48
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
CRACR2A Q9BSW2 1/20 0.42
NAPRT Q6XQN6 1/20 0.42
SLC16A3 O15427 1/20 0.42
POLB P06746 1/20 0.42
TSHR P16473 1/20 0.42
NPSR1 Q6W5P4 2/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
ALDH1A1 P00352 1/20 0.41
PKM P14618 1/20 0.41
P2RX7 Q99572 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22637715 1.00 SORT1 (0.57) SORT1GRNMARS1KLKB1CYP1A2
SCHEMBL4134838 0.87 GRN (0.74) SORT1GRNKLKB1POLBTSHR
SCHEMBL22637502 0.84 GRN (0.59) SORT1GRNMARS1KLKB1NPSR1
SCHEMBL22637209 0.84 SMN1; SMN2 (0.52) SORT1GRNCYP1A2CYP3A4CYP2D6
SCHEMBL27727953 0.77 GRN (0.47) SORT1GRNKLKB1CYP1A2CYP3A4
SCHEMBL29008667 0.76 GRN (0.76) SORT1GRNKLKB1POLBTSHR
SCHEMBL2688186 0.75 GRN (0.57) SORT1GRNKLKB1NPSR1GAA
SCHEMBL3069753 0.73 GRN (1.00) SORT1GRNCYP1A2CYP2D6CYP2C9
SCHEMBL4253961 0.72 PTGS2 (0.51) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL19779588 0.72 CCR9 (0.51) SORT1GRNKLKB1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114269340-A KCNT1 inhibitors and methods of use 普拉克西斯精密药物股份有限公司 2022-04-01 CN disclosed