SCHEMBL29480975

SCHEMBL29480975

COC(=O)c1cccc(Br)c1C(=O)C(C)C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F2R P25116 1/20 0.43
LMNA P02545 2/20 0.43
TSHR P16473 1/20 0.43
ALDH1A1 P00352 3/20 0.42
CFTR P13569 1/20 0.42
HSD17B10 Q99714 1/20 0.42
SLC6A3 Q01959 1/20 0.42
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
CA9 Q16790 2/20 0.42
CA12 O43570 1/20 0.42
CA7 P43166 1/20 0.42
CA14 Q9ULX7 1/20 0.42
CA5A P35218 1/20 0.41
KDM4E B2RXH2 3/20 0.41
ATM Q13315 2/20 0.41
POLB P06746 1/20 0.41
KMT2A Q03164 5/20 0.41
MEN1 O00255 2/20 0.41
CYP1A2 P05177 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30368137 0.84 CA1 (0.53) LMNATSHRALDH1A1CFTRHSD17B10
SCHEMBL1962462 0.84 CA1 (0.53) LMNATSHRALDH1A1CFTRHSD17B10
SCHEMBL29480920 0.83 TSHR (0.53) F2RLMNATSHRALDH1A1HSD17B10
SCHEMBL29401587 0.81 PRNP (0.44) F2RALDH1A1HSD17B10CA1CA2
SCHEMBL24254622 0.80 FFAR1 (0.43) F2RTSHRALDH1A1CA1CA2
SCHEMBL31582602 0.79 LMNA (0.44) LMNATSHRALDH1A1CFTRHSD17B10
SCHEMBL851838 0.77 CA1 (0.61) LMNATSHRALDH1A1CFTRHSD17B10
SCHEMBL10161076 0.75 TSHR (0.57) LMNATSHRALDH1A1CFTRHSD17B10
SCHEMBL29279663 0.75 TSHR (0.52) LMNATSHRALDH1A1CFTRHSD17B10
SCHEMBL31347202 0.75 TSHR (0.44) LMNATSHRALDH1A1CFTRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114174278-A Dihydroorotate dehydrogenase inhibitors 詹森生物科技公司 2022-03-11 CN disclosed