SCHEMBL29482199

SCHEMBL29482199

N#Cc1ccccc1C(=O)N1CCOCC1

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.58
GAA P10253 2/20 0.57
SMN1; SMN2 Q16637 2/20 0.57
ALDH1A1 P00352 4/20 0.56
HSD11B1 P28845 1/20 0.55
TSHR P16473 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
TP53 P04637 1/20 0.52
KMT2A Q03164 2/20 0.51
HTT P42858 1/20 0.50
PKM P14618 1/20 0.49
MEN1 O00255 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7276196 0.86 GAA (0.59) CNR1GAASMN1; SMN2ALDH1A1TSHR
SCHEMBL4599304 0.85 HSD11B1 (0.59) SMN1; SMN2ALDH1A1HSD11B1TSHRKMT2A
SCHEMBL7121916 0.83 SMN1; SMN2 (0.77) GAASMN1; SMN2ALDH1A1TSHRNPSR1
SCHEMBL3092100 0.83 HSD11B1 (0.56) CNR1ALDH1A1HSD11B1TSHRKMT2A
SCHEMBL28812724 0.81 RXFP1 (0.60) ALDH1A1HSD11B1
SCHEMBL24363913 0.80 CNR1 (0.54) CNR1GAASMN1; SMN2ALDH1A1TSHR
SCHEMBL19657125 0.80 CNR1 (0.54) CNR1ALDH1A1TSHRTP53HTT
SCHEMBL1447674 0.80 KDM4E (0.63) CNR1GAASMN1; SMN2TSHRKMT2A
SCHEMBL30367909 0.79 HSD11B1 (0.56) CNR1SMN1; SMN2ALDH1A1HSD11B1TSHR
(2-Aminophenyl)(Morpholino)Methanone SCHEMBL30988542 0.79 GAA (0.62) GAASMN1; SMN2ALDH1A1TSHRNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3218375-B1 SUBSTITUTED PYRROLOPYRDINES AS INHIBITORS OF BROMODOMAIN GENENTECH INC (US) 2022-04-27 EP claimed