SCHEMBL2948723

SCHEMBL2948723

CCCCn1cnc2c(=O)n(C)c(=O)[nH]c21

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.53
KDM4E B2RXH2 6/20 0.50
ALDH1A1 P00352 6/20 0.50
HPGD P15428 4/20 0.50
HSD17B10 Q99714 2/20 0.50
KMT2A Q03164 3/20 0.49
PKM P14618 1/20 0.48
MEN1 O00255 2/20 0.48
ADORA2A P29274 3/20 0.46
PDE4A P27815 1/20 0.46
PDE4B Q07343 1/20 0.46
PDE4C Q08493 1/20 0.46
PDE4D Q08499 1/20 0.46
NPC1 O15118 2/20 0.44
RAB9A P51151 1/20 0.43
CYP2C9 P11712 1/20 0.43
BRD4 O60885 1/20 0.43
BRD2 P25440 1/20 0.43
BRD3 Q15059 1/20 0.43
BRDT Q58F21 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10432471 0.83 HSD17B10 (0.49) GAAKDM4EALDH1A1HPGDHSD17B10
SCHEMBL7367989 0.81 ALDH1A1 (0.46) GAAKDM4EALDH1A1HPGDHSD17B10
SCHEMBL6233163 0.78 PNP (0.58) GAAKDM4EALDH1A1HPGDKMT2A
SCHEMBL9885890 0.77 KMT2A (0.47) GAAKDM4EALDH1A1HPGDKMT2A
SCHEMBL9885887 0.77 KMT2A (0.47) GAAKDM4EALDH1A1HPGDKMT2A
SCHEMBL9199287 0.76 LMNA (0.40) GAAKDM4EALDH1A1HPGDHSD17B10
SCHEMBL515776 0.76 ALDH1A1 (0.54) GAAKDM4EALDH1A1HPGDHSD17B10
SCHEMBL9845193 0.75 GAA (0.59) GAAKDM4EALDH1A1HPGDHSD17B10
SCHEMBL13728723 0.75 GAA (0.59) GAAKDM4EALDH1A1HPGDHSD17B10
SCHEMBL27193125 0.73 PDE4A (0.55) KDM4EALDH1A1HPGDHSD17B10KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4401833-A1 GPR52 MODULATOR COMPOUNDS Nxera Pharma UK Limited (GB) 2024-07-24 EP disclosed
EP-4204408-A1 GPR52 MODULATOR COMPOUNDS Heptares Therapeutics Limited (GB) 2023-07-05 EP disclosed
WO-2023041909-A1 GPR52 MODULATOR COMPOUNDS HEPTARES THERAPEUTICS LIMITED (GB) 2023-03-23 WO disclosed
WO-2022043714-A1 GPR52 MODULATOR COMPOUNDS HEPTARES THERAPEUTICS LIMITED (GB) 2022-03-03 WO disclosed
CN-111467345-A Method for inhibiting growth and metastasis of solid tumor cells and special pharmaceutical composition 天津市人民医院 2020-07-31 CN disclosed
CN-110499285-A Application of the ALPL gene in the product of preparation prevention and/or treatment low alkalinity phosphatase disease XIAN TISSUE ENGINEERING AND REGENERATIVE MEDICINE RES INSTITUTE 2019-11-26 CN disclosed
CN-109988746-A A kind of mescenchymal stem cell adipogenic induction differentiation method 上海葆年生物科技有限公司 2019-07-09 CN disclosed
CN-109714962-A Systems and methods for culturing cells in vitro 耶路撒冷希伯来大学的益生研究开发有限公司 2019-05-03 CN disclosed
CN-105343894-B The recombination mescenchymal stem cell of efficient secretion prostaglandin E2 (PGE2) and its application 中国人民解放军军事医学科学院基础医学研究所 2019-01-29 CN disclosed
CN-109182256-A A kind of spotted maigre Preadipocyte In Vitro be separately cultured and its abductive approach 浙江省海洋水产研究所 2019-01-11 CN disclosed
CN-108192856-A A kind of method for efficiently separating and cultivating the primary melanocyte of people 山东大学 2018-06-22 CN disclosed
CN-107864627-A Include the method and composition of adhering substrate cell 普拉里斯坦有限公司 2018-03-30 CN disclosed
CN-107849533-A Use of mesenchymal stem cells for the treatment of osteoarthritis 洪士杰 2018-03-27 CN disclosed
CN-104277112-B Long-acting hypoglycemic fusion protein 嘉和生物药业有限公司 2018-01-26 CN disclosed
CN-107106613-A Composition comprising stem cell-derived exosomes for adipogenic differentiation induction, adipose tissue regeneration, skin whitening or wrinkle improvement 胞外体干细胞株式会社 2017-08-29 CN disclosed
CN-106754664-A It is a kind of to induce the culture medium that break up into fat of Skeletal Muscle derived stem cells and its apply and into fat differentiation method 广州赛莱拉干细胞科技股份有限公司 2017-05-31 CN disclosed
CN-106508892-A Umbilical cord tissue cryopreservation solution and cryopreservation method 广州赛莱拉干细胞科技股份有限公司 2017-03-22 CN disclosed
CN-106381283-A Adipogenesis induction culture medium and adipogenic differentiation method 广州赛莱拉干细胞科技股份有限公司 2017-02-08 CN disclosed
WO-2014205081-A1 PHARMACEUTICAL FORMULATIONS OF XANTHINE OR XANTHINE DERIVATIVES, AND THEIR USE IMPRIMIS PHARMACEUTICALS INC. (US) 2014-12-24 WO disclosed
EP-1735278-B1 HISTAMINE H3 RECEPTOR AGENTS, PREPARATION AND THERAPEUTIC USES LILLY CO ELI (US) 2010-01-06 EP disclosed