SCHEMBL29488256

SCHEMBL29488256

Nc1ccc2nc(C(=O)c3cccc(C(F)(F)F)c3)[nH]c(=O)c2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 2/20 0.46
SRD5A2 P31213 1/20 0.45
CNR2 P34972 2/20 0.45
ABCG2 Q9UNQ0 2/20 0.44
PTGS1 P23219 3/20 0.44
KDM4E B2RXH2 2/20 0.43
TOP2A P11388 1/20 0.43
TOP2B Q02880 1/20 0.43
HTT P42858 1/20 0.43
CES2 O00748 1/20 0.42
ALDH1A1 P00352 2/20 0.41
HSD17B10 Q99714 2/20 0.41
MEN1 O00255 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
MAPT P10636 1/20 0.41
ADORA1 P30542 1/20 0.41
KMT2A Q03164 1/20 0.41
BRD4 O60885 1/20 0.41
HPGD P15428 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28738669 1.00 MGLL (0.46) MGLLSRD5A2CNR2ABCG2PTGS1
SCHEMBL28738679 0.84 TOP2A (0.54) TOP2ATOP2BHTTALDH1A1MEN1
SCHEMBL29488266 0.83 ABCG2 (0.48) MGLLABCG2MEN1MAPTKMT2A
SCHEMBL28738683 0.83 ABCG2 (0.48) MGLLABCG2MEN1MAPTKMT2A
SCHEMBL29488269 0.80 MAPT (0.45) MGLLHTTALDH1A1MAPT
SCHEMBL28308601 0.80 MAPT (0.45) MGLLHTTALDH1A1MAPT
SCHEMBL29488268 0.80 MAPT (0.45) MGLLHTTALDH1A1MAPT
SCHEMBL29488270 0.79 XDH (0.50) KDM4ETOP2ATOP2BCES2ALDH1A1
SCHEMBL28738673 0.79 XDH (0.50) KDM4ETOP2ATOP2BCES2ALDH1A1
SCHEMBL17786457 0.77 TNKS (0.53) ABCG2KDM4EHTTALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109897008-B 2-benzoyl-6-amino-4 (3H) -quinazolinone derivative and synthesis method and application thereof 中南大学 2022-05-03 CN disclosed