SCHEMBL29488258

SCHEMBL29488258

COc1ccc(C(=O)c2nc3ccc(N)cc3c(=O)[nH]2)cc1OC

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.52
TSHR P16473 2/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
MEN1 O00255 5/20 0.43
KMT2A Q03164 5/20 0.43
POLB P06746 3/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
APAF1 O14727 1/20 0.43
NSD2 O96028 1/20 0.43
CASP3 P42574 1/20 0.43
SENP8 Q96LD8 1/20 0.43
SENP7 Q9BQF6 1/20 0.43
SENP6 Q9GZR1 1/20 0.43
ESR1 P03372 1/20 0.43
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28738687 1.00 BRD4 (0.52) BRD4TSHRCYP1A2CYP3A4CYP2C9
SCHEMBL28738700 0.83 ALDH1A1 (0.52) BRD4TSHRCYP1A2CYP3A4CYP2C9
SCHEMBL29488267 0.83 ALDH1A1 (0.52) BRD4TSHRCYP1A2CYP3A4CYP2C9
SCHEMBL28738695 0.82 BRD4 (0.51) BRD4MEN1KMT2APOLBSMN1; SMN2
SCHEMBL28738679 0.80 TOP2A (0.54) BRD4TSHRMEN1KMT2APOLB
SCHEMBL29488265 0.79 MAPT (0.46) BRD4TSHRMEN1KMT2APOLB
SCHEMBL29488264 0.79 MAPT (0.46) BRD4TSHRMEN1KMT2APOLB
SCHEMBL28308709 0.79 MAPT (0.46) BRD4TSHRMEN1KMT2APOLB
SCHEMBL28738662 0.77 BRD4 (0.46) BRD4MEN1KMT2ANPC1TOP2A
SCHEMBL17786541 0.76 GUSB (0.71) CYP1A2MEN1KMT2APOLBCASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109897008-B 2-benzoyl-6-amino-4 (3H) -quinazolinone derivative and synthesis method and application thereof 中南大学 2022-05-03 CN disclosed