SCHEMBL29498705

SCHEMBL29498705

FC(F)c1ccccc1Br

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.42
TDO2 P48775 1/20 0.42
ALDH1A1 P00352 5/20 0.38
HTT P42858 1/20 0.36
MAPK1 P28482 1/20 0.35
OPRL1 P41146 2/20 0.34
CYP2C19 P33261 3/20 0.33
CYP3A4 P08684 1/20 0.33
ALOX15 P16050 1/20 0.33
CA1 P00915 2/20 0.32
CA2 P00918 2/20 0.32
CA4 P22748 1/20 0.32
CA6 P23280 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
CFTR P13569 2/20 0.32
OPRM1 P35372 1/20 0.32
OPRD1 P41143 1/20 0.32
OPRK1 P41145 1/20 0.32
CYP2C9 P11712 2/20 0.31
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL183025 1.00 IDO1 (0.42) IDO1TDO2ALDH1A1HTTMAPK1
SCHEMBL23430140 0.82 HTR3E (0.33) IDO1TDO2ALDH1A1HTTOPRL1
SCHEMBL15973428 0.79 HTT (0.42) IDO1TDO2ALDH1A1HTTMAPK1
SCHEMBL1538924 0.78 GABRA1 (0.35) IDO1TDO2ALDH1A1HTTMAPK1
SCHEMBL29861488 0.77 IDO1 (0.31) IDO1TDO2
SCHEMBL29525404 0.77 KDM1A (0.31) IDO1TDO2
SCHEMBL23326396 0.77 IDO1 (0.31) IDO1TDO2
SCHEMBL16636835 0.77 KDM1A (0.31) IDO1TDO2
SCHEMBL4087851 0.77 IDO1 (0.45) IDO1TDO2ALDH1A1HTTMAPK1
SCHEMBL21132602 0.75 ALDH1A1 (0.37) ALDH1A1MAPK1CYP3A4CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114524776-B Tetrazole compound and application thereof 中国科学院广州生物医药与健康研究院 2024-12-13 CN disclosed
EP-4380560-A1 LPAR1 ANTAGONISTS AND USES THEREOF Contineum Therapeutics, Inc. (US) 2024-06-12 EP disclosed
CN-118164961-A 4-Methylsulfonyl substituted piperidine urea compounds for the treatment of Dilated Cardiomyopathy (DCM) 迈奥卡迪亚公司 2024-06-11 CN disclosed
CN-111393414-B 4-Methylsulfonyl substituted piperidine urea compounds for the treatment of Dilated Cardiomyopathy (DCM) 迈奥卡迪亚公司 2024-05-07 CN disclosed
WO-2023122093-A1 REV-ERB AGONISTS FOR TH17-MEDIATED INFLAMMATORY DISORDERS UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2023-06-29 WO disclosed
CN-115989228-A Heterocyclic compounds 豪夫迈·罗氏有限公司 2023-04-18 CN disclosed
CN-115916756-A Sulfone derivative 豪夫迈·罗氏有限公司 2023-04-04 CN disclosed
WO-2023014908-A1 LPAR1 ANTAGONISTS AND USES THEREOF Pipeline Therapeutics, Inc. (US) 2023-02-09 WO disclosed
CN-114702495-A Purinones as ubiquitin-specific protease 1 inhibitors 福马治疗有限公司 2022-07-05 CN disclosed
CN-110248940-B Aryl hydrocarbon receptor (AhR) modulator compounds 菲尼克斯药品股份公司 2022-07-01 CN disclosed
CN-109689642-B Monocyclic heteroaryl substituted compounds 百时美施贵宝公司 2022-04-12 CN disclosed
CN-108473495-B Purinones as ubiquitin-specific protease 1 inhibitors 福马治疗有限公司 2022-04-12 CN disclosed