SCHEMBL29501775

SCHEMBL29501775

COC(=O)[C@H](CCC(=O)OCc1ccccc1)NC(=O)[C@H](CCCNC(=N)NS(=O)(=O)c1c(C)c(C)c2c(c1C)CC(C)(C)O2)NC(=O)[C@H](CCCCNC(=O)OCc1ccccc1)NC(=O)OC(C)(C)C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KLK7 P49862 2/20 0.44
KLK5 Q9Y337 2/20 0.44
MAPT P10636 1/20 0.40
ITGB3 P05106 1/20 0.39
ITGA2B P08514 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
SIRT2 Q8IXJ6 1/20 0.37
SIRT1 Q96EB6 1/20 0.37
SIRT3 Q9NTG7 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
TLR2 O60603 1/20 0.37
TLR1 Q15399 1/20 0.37
PSMB8 P28062 1/20 0.36
PSMB9 P28065 1/20 0.36
PSMB5 P28074 1/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29501799 0.93 KLK7 (0.47) KLK7KLK5MAPTITGB3ITGA2B
SCHEMBL31058627 0.87 PLG (0.32) KLK7KLK5CA1CA2TDP1
SCHEMBL29501759 0.85 ITGB3 (0.37) KLK7KLK5ITGB3ITGA2B
SCHEMBL22834294 0.85 ITGB3 (0.37) KLK7KLK5ITGB3ITGA2B
SCHEMBL22834296 0.85 ITGB3 (0.37) KLK7KLK5ITGB3ITGA2B
SCHEMBL30134454 0.85 ITGB3 (0.42) ITGB3SIRT2SIRT1SIRT3FOLH1
SCHEMBL12637855 0.83 KLK7 (0.39) KLK7KLK5MAPTITGB3ITGA2B
SCHEMBL31058628 0.83 ALDH1A1 (0.37) KLK7KLK5ITGB3ITGA2BCA1
SCHEMBL31758414 0.82 PTGER4 (0.41) SIRT2SIRT1SIRT3MEN1ALDH1A1
SCHEMBL29401366 0.82 ITGB3 (0.44) ITGB3SIRT2SIRT1FOLH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3989997-A1 COMPOUNDS AND METHODS FOR TREATING CANCER, VIRAL INFECTIONS, AND ALLERGIC CONDITIONS Washington University (US) 2022-05-04 EP disclosed