SCHEMBL29501799

SCHEMBL29501799

Cc1c(C)c(S(=O)(=O)NC(=N)NCCC[C@H](NC(=O)[C@H](CCCCNC(=O)OCc2ccccc2)NC(=O)OC(C)(C)C)C(=O)O)c(C)c2c1OC(C)(C)C2

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KLK7 P49862 2/20 0.47
KLK5 Q9Y337 2/20 0.47
MAPT P10636 1/20 0.43
ITGB3 P05106 1/20 0.41
ITGA2B P08514 1/20 0.41
MMP2 P08253 2/20 0.40
MMP9 P14780 2/20 0.40
CPB1 P15086 1/20 0.40
CPB2 Q96IY4 1/20 0.40
FOLH1 Q04609 2/20 0.40
ALDH1A1 P00352 1/20 0.40
TSHR P16473 1/20 0.40
TDP1 Q9NUW8 1/20 0.39
PTGER4 P35408 1/20 0.39
PSMB8 P28062 1/20 0.39
PSMB9 P28065 1/20 0.39
PSMB5 P28074 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29501775 0.93 KLK7 (0.44) KLK7KLK5MAPTITGB3ITGA2B
SCHEMBL30134454 0.92 ITGB3 (0.42) ITGB3MMP2MMP9CPB1CPB2
SCHEMBL31058628 0.90 ALDH1A1 (0.37) KLK7KLK5ITGB3ITGA2BMMP9
SCHEMBL29398651 0.90 ITGB3 (0.44) ITGB3MMP2MMP9FOLH1
SCHEMBL29401366 0.90 ITGB3 (0.44) ITGB3MMP2MMP9FOLH1
SCHEMBL16893643 0.88 ALDH1A1 (0.41) KLK7KLK5ITGB3ITGA2BALDH1A1
SCHEMBL30918351 0.88 ALDH1A1 (0.35) KLK7KLK5ALDH1A1TSHR
SCHEMBL20561238 0.88 ALDH1A1 (0.39) KLK7KLK5ITGB3ITGA2BALDH1A1
SCHEMBL29401007 0.88 ALDH1A1 (0.39) KLK7KLK5ITGB3ITGA2BALDH1A1
SCHEMBL15407157 0.88 ALDH1A1 (0.39) KLK7KLK5ITGB3ITGA2BALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3989997-A1 COMPOUNDS AND METHODS FOR TREATING CANCER, VIRAL INFECTIONS, AND ALLERGIC CONDITIONS Washington University (US) 2022-05-04 EP disclosed