SCHEMBL29503148

SCHEMBL29503148

CP(C)(=O)c1cccc(C(N)=O)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 11/20 0.55
TSHR P16473 2/20 0.45
POLB P06746 1/20 0.45
CYP3A4 P08684 1/20 0.45
MAPT P10636 1/20 0.45
CYP2C19 P33261 1/20 0.45
RECQL P46063 1/20 0.45
BLM P54132 1/20 0.45
PMP22 Q01453 1/20 0.45
HSD17B10 Q99714 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
PARP10 Q53GL7 4/20 0.45
PARP15 Q460N3 2/20 0.45
PARP14 Q460N5 2/20 0.43
TNKS O95271 1/20 0.43
TNKS2 Q9H2K2 1/20 0.43
PARP2 Q9UGN5 1/20 0.43
BAZ2B Q9UIF8 1/20 0.41
BAZ2A Q9UIF9 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26185623 0.82 CA12 (0.50) TSHRPOLBMAPTRECQLBLM
SCHEMBL29700464 0.82 CA12 (0.50) TSHRPOLBMAPTRECQLBLM
SCHEMBL30574149 0.80 PARP1 (0.54) PARP1TSHRPOLBCYP3A4MAPT
SCHEMBL30223402 0.79 HDAC8 (0.59) TSHRPOLBL3MBTL1MEN1KMT2A
SCHEMBL30223420 0.79 HDAC8 (0.59) TSHRPOLBL3MBTL1MEN1KMT2A
SCHEMBL24478812 0.78 RAB9A (0.53) TSHRPOLBCYP3A4MAPTCYP2C19
SCHEMBL30184543 0.78 KMT2A (0.44) TDP1L3MBTL1MEN1KMT2A
SCHEMBL31317830 0.78 RAB9A (0.53) TSHRPOLBCYP3A4MAPTCYP2C19
SCHEMBL36694 0.76 PARP1 (0.73) PARP1TSHRPOLBCYP3A4MAPT
SCHEMBL31021028 0.76 PARP1 (0.73) PARP1TSHRPOLBCYP3A4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111601790-B Heteroaryl compounds as protein kinase inhibitors 福建海西新药创制股份有限公司 2023-03-31 CN claimed
CN-115697993-B Pyrimidine compounds as AXL inhibitors 南京正大天晴制药有限公司 2024-12-10 CN disclosed
CN-111601790-B Heteroaryl compounds as protein kinase inhibitors 福建海西新药创制股份有限公司 2023-03-31 CN disclosed
CN-115697993-A Pyrimidines as AXL inhibitors 南京正大天晴制药有限公司 2023-02-03 CN disclosed