SCHEMBL29520358

SCHEMBL29520358

Clc1ncc(Cl)c(-c2nccc3ccccc23)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RPS6KA5 O75582 2/20 0.48
NPY5R Q15761 1/20 0.46
KDM4E B2RXH2 4/20 0.43
NPC1 O15118 4/20 0.43
RAB9A P51151 4/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
GPR55 Q9Y2T6 1/20 0.43
MAPT P10636 5/20 0.43
KMT2A Q03164 2/20 0.43
GLA P06280 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
CYP2A6 P11509 3/20 0.42
PLAU P00749 2/20 0.42
F12 P00748 1/20 0.42
NCF1 P14598 1/20 0.42
NOS3 P29474 1/20 0.42
NOS1 P29475 1/20 0.42
NOS2 P35228 1/20 0.42
BACE1 P56817 1/20 0.42
MAPK1 P28482 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL266030 0.84 CYP2A6 (0.47) RPS6KA5NPY5RKDM4ENPC1RAB9A
SCHEMBL29923403 0.80 PLAU (0.60) NPY5RKDM4ENPC1RAB9AL3MBTL1
SCHEMBL199273 0.80 PLAU (0.60) NPY5RKDM4ENPC1RAB9AL3MBTL1
SCHEMBL30522769 0.78 PLAU (0.58) NPY5RKDM4ENPC1RAB9AL3MBTL1
SCHEMBL31175962 0.74 CYP2A6 (0.52) NPY5RKDM4ENPC1RAB9AL3MBTL1
SCHEMBL28252191 0.74 HTR1A (0.51) NPY5RKDM4ENPC1RAB9AL3MBTL1
SCHEMBL29651118 0.72 RPS6KA5 (0.50) RPS6KA5CYP3A4CYP1A2CYP2C19
SCHEMBL28743633 0.72 RPS6KA5 (0.50) RPS6KA5CYP3A4CYP1A2CYP2C19
SCHEMBL12223316 0.72 PLAU (0.56) NPY5RKDM4ENPC1RAB9AL3MBTL1
SCHEMBL13978866 0.72 PLAU (0.56) NPY5RKDM4ENPC1RAB9AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022063140-A1 PYRIMIDINE AND PYRIDINE DERIVATIVES AS HPK1 MODULATOR AND METHODS USING SAME SHENZHEN IONOVA LIFE SCIENCE CO., LTD. (CN) 2022-03-31 WO disclosed