SCHEMBL29520494

SCHEMBL29520494

CC(C)=C1C(c2ccccc2)=NC(C(C)(C)C)=Nc2ccc(C(C)C)cc21

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.38
CYP1A2 P05177 1/20 0.34
POLB P06746 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
PTPN5 P54829 1/20 0.32
IDO1 P14902 1/20 0.32
METAP2 P50579 1/20 0.32
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29520545 0.84 MAPT (0.42) MAPTCYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL29520664 0.83 CHRM1 (0.39) MAPTCYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL29520576 0.83 IDO1 (0.31) IDO1
SCHEMBL29521036 0.83 CYP2C9 (0.36) MAPTCYP2C9CYP2C19IDO1LMNA
SCHEMBL28500399 0.81 MAPT (0.43) MAPTLMNA
SCHEMBL29520828 0.81 MAPT (0.45) MAPTCYP1A2CYP2C9CYP2C19LMNA
SCHEMBL29520554 0.81 CHRM1 (0.37)
SCHEMBL29520737 0.80 IDO1 (0.40) MAPTIDO1LMNA
SCHEMBL29409248 0.78 NPC1 (0.36) MAPTLMNA
SCHEMBL29520778 0.77 CHRM1 (0.37) LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112174901-B Synthesis method and anticancer activity of 1, 3-benzodiazepine compound 河南师范大学 2022-02-08 CN disclosed