SCHEMBL29522657

SCHEMBL29522657

NC(=O)c1ccc2cnccc2c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.62
LCK P06239 1/20 0.56
SMYD3 Q9H7B4 2/20 0.54
CYP3A4 P08684 5/20 0.51
F7 P08709 1/20 0.48
F3 P13726 1/20 0.48
SARM1 Q6SZW1 1/20 0.48
SIRT2 Q8IXJ6 1/20 0.48
SIRT6 Q8N6T7 1/20 0.48
SIRT1 Q96EB6 1/20 0.48
SIRT3 Q9NTG7 1/20 0.48
SIRT5 Q9NXA8 1/20 0.48
SIRT4 Q9Y6E7 1/20 0.48
HIPK2 Q9H2X6 1/20 0.47
CHEK1 O14757 1/20 0.47
AURKA O14965 1/20 0.47
DAPK3 O43293 1/20 0.47
PRKD3 O94806 1/20 0.47
MAP4K4 O95819 1/20 0.47
PAK4 O96013 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4280154 1.00 AR (0.62) ARLCKSMYD3CYP3A4F7
SCHEMBL6648425 0.93 AR (0.55) ARLCKSMYD3CYP3A4F7
SCHEMBL29972759 0.93 AR (0.55) ARLCKSMYD3CYP3A4F7
SCHEMBL18318801 0.86 AR (0.64) ARCYP3A4MAP4K4MKNK1MKNK2
SCHEMBL113378 0.83 SMYD3 (0.55) ARSMYD3CYP3A4HIPK2IMPDH2
SCHEMBL29489099 0.83 SMYD3 (0.55) ARSMYD3CYP3A4HIPK2IMPDH2
SCHEMBL2363489 0.82 LCK (0.78) LCKPLAUKDM4E
SCHEMBL12765931 0.81 SMYD3 (0.50) ARSMYD3CYP3A4HIPK2IMPDH2
SCHEMBL3126130 0.81 IMPDH2 (0.53) ARSMYD3CYP3A4HIPK2IMPDH2
Hydrochloric Acid SCHEMBL7557776 0.81 SMYD3 (0.54) ARSMYD3CYP3A4HIPK2IMPDH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3536685-B1 BICYCLIC-FUSED HETEROARYL OR ARYL COMPOUNDS AND THEIR USE AS IRAK4 INHIBITORS PFIZER (US) 2022-02-16 EP claimed
WO-2024032715-A1 HYDRAZIDE COMPOUND AND PREPARATION METHOD THEREFOR AND USE THEREOF 深圳微芯生物科技股份有限公司 2024-02-15 WO disclosed
EP-3640242-B1 ROCK-INHIBITING COMPOUND AND USES THEREOF HITGEN LTD (CN) 2023-04-19 EP disclosed
EP-4125900-A1 METHODS OF TREATING CORONAVIRUS DISEASE 2019 Pfizer Inc. (US) 2023-02-08 EP disclosed
CN-114423757-A Tricyclic heteroaryl compounds useful as IRAK4 inhibitors 百时美施贵宝公司 2022-04-29 CN disclosed