Cloxacillin

Cloxacillin

SCHEMBL2953

Cc1onc(-c2ccccc2Cl)c1C(=O)N[C@@H]1C(=O)N2[C@@H]1SC(C)(C)[C@@H]2C(=O)O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

mecApbp2pbp4pbpApbpF

The experimentally established mechanism targets of Cloxacillin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ABCB11 O95342 3/20 1.00
LMNA P02545 4/20 0.84
HPGD P15428 3/20 0.84
CYP1A2 P05177 1/20 0.79
KMT2A Q03164 2/20 0.71
MEN1 O00255 1/20 0.71
TDP1 Q9NUW8 1/20 0.71
SLCO1B3 Q9NPD5 1/20 0.70
SLCO1B1 Q9Y6L6 1/20 0.70
ALDH1A1 P00352 1/20 0.68
SMN1; SMN2 Q16637 1/20 0.68
PTGS1 P23219 1/20 0.55
PDE3A Q14432 1/20 0.55
HRH1 P35367 1/20 0.51
SLC22A8 Q8TCC7 1/20 0.51
CYP2C19 P33261 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cloxacillin SCHEMBL11404593 1.00 ABCB11 (1.00) ABCB11LMNAHPGDCYP1A2KMT2A
Cloxacillin SCHEMBL11404577 1.00 ABCB11 (1.00) ABCB11LMNAHPGDCYP1A2KMT2A
Cloxacillin SCHEMBL16333855 1.00 ABCB11 (1.00) ABCB11LMNAHPGDCYP1A2KMT2A
Cloxacillin SCHEMBL1625107 1.00 ABCB11 (1.00) ABCB11LMNAHPGDCYP1A2KMT2A
Cloxacillin SCHEMBL31229061 1.00 ABCB11 (1.00) ABCB11LMNAHPGDCYP1A2KMT2A
Cloxacillin SCHEMBL8728823 1.00 ABCB11 (1.00) ABCB11LMNAHPGDCYP1A2KMT2A
Cloxacillin SCHEMBL11404582 1.00 ABCB11 (1.00) ABCB11LMNAHPGDCYP1A2KMT2A
Cloxacillin SCHEMBL41014 0.99 ABCB11 (0.98) ABCB11LMNAHPGDCYP1A2KMT2A
Cloxacillin SCHEMBL28547421 0.99 ABCB11 (0.98) ABCB11LMNAHPGDCYP1A2KMT2A
Cloxacillin SCHEMBL5550210 0.98 ABCB11 (0.97) ABCB11LMNAHPGDCYP1A2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 25926 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12637481-B2 Boronic acid derivatives and therapeutic uses thereof QPEX BIOPHARMA, INC. (US) 2026-05-26 US claimed
WO-2026106917-A1 EDIBLE TRANSMUCOSAL DRUG DELIVERY METHOD USING AN INTERMEDIATE CAPSULE AS A TEMPORARY VESSEL BioPhysics Pharma, Inc. (US) 2026-05-21 WO claimed
WO-2026104587-A1 CYCLIC BORONIC ACID ESTERS USEFUL AS ADJUVANTS IN THE TREATMENT OF BACTERIAL INFECTIONS ADJUTEC PHARMA AS (NO) 2026-05-21 WO claimed
EP-4736859-A1 ANTIBIOTIC COMPOSITIONS University of Galway (IE) 2026-05-06 EP claimed
US-20260108619-A1 CONJUGATION LINKERS, CELL BINDING MOLECULE-DRUG CONJUGATES CONTAINING THE LINKERS, METHODS OF MAKING AND USES SUCH CONJUGATES WITH THE LINKERS HANGZHOU DAC BIOTECH CO., LTD. (CN) 2026-04-23 US claimed
US-12605345-B2 Transdermal drug delivery system BioPhysics Pharma, Inc. (US) 2026-04-21 US claimed
EP-4724049-A1 MODIFIED RELEASE FILL COMPOSITIONS FOR DOSAGE FORMS AND METHODS OF PREPARATION AND USE THEREOF Catalent Ontario Limited (CA) 2026-04-15 EP claimed
US-12594365-B2 Ionic compounds for medical device applications BECTON, DICKINSON AND COMPANY (US) 2026-04-07 US claimed
US-20260091089-A1 Pyocyanine Demethylases and related Phenazine Degrading Agents Compositions, Methods and Systems for Interfering with Viability of Bacteria CALIFORNIA INST OF TECHN (US) 2026-04-02 US claimed
US-20260091127-A1 JANUS PARTICLE-EMBEDDED MATERIALS FOR ANTIMICROBIAL APPLICATIONS UNIV INDIANA TRUSTEES (US) 2026-04-02 US claimed
US-4302447-A Pharmaceutical and dietary composition EFAMOL LIMITED (GB) 1981-11-24 US claimed
EP-0003407-B1 PHARMACEUTICAL AND DIETARY COMPOSITION COMPRISING GAMMA-LINOLENIC ACIDS EFAMOL LIMITED (GB) 1981-09-30 EP claimed
US-4283400-A Medicated animal feed based on liver meal BAYER AKTIENGESELLSCHAFT (DE) 1981-08-11 US claimed
US-4273763-A TREATMENT OF SCHIZOPHRENIA WITH B-LACTAM ANTIBIOTICS EFAMOL LIMITED (GB) 1981-06-16 US claimed
EP-0029668-A1 Pharmaceutical injectable composition and two-pack container for said composition BEECHAM GROUP PLC (GB) 1981-06-03 EP claimed
US-4239745-A INCUBATION WITH TAGGED ANTIBIOTIC AND ANTIBIOTIC SENSITIVE CELLS PENICILLIN ASSAYS, INC. (US) 1980-12-16 US claimed
US-4217274-A Methoxyethoxymethyl esters of penicillins BRISTOL-MYERS COMPANY (US) 1980-08-12 US claimed
US-4199566-A DERIVATIVES OF PENICILLANIC ACID TOYAMA CHEMICAL COMPANY, LIMITED (JP) 1980-04-22 US claimed
EP-0004770-A2 Pharmaceutical and dietary composition comprising gamma-linolenic acids EFAMOL LIMITED (GB) 1979-10-17 EP claimed
US-4145429-A VEGETALBE OIL, CLAY, ANTIBIOTIC BEECHAM GROUP LIMITED (GB) 1979-03-20 US claimed