SCHEMBL2953053

SCHEMBL2953053

Nc1nc(N)c2nc(-c3ccc(N4CCOCC4)cn3)[nH]c2n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADK P55263 1/20 0.42
DHFR P00374 2/20 0.42
CBFB Q13951 1/20 0.42
XDH P47989 1/20 0.40
JAK2 O60674 3/20 0.39
JAK1 P23458 3/20 0.39
TYK2 P29597 3/20 0.39
JAK3 P52333 3/20 0.39
TBK1 Q9UHD2 1/20 0.39
POLB P06746 1/20 0.38
IGF1R P08069 2/20 0.38
CDK1 P06493 1/20 0.38
CDK2 P24941 1/20 0.38
ATR Q13535 1/20 0.37
NOS1 P29475 1/20 0.37
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37
MAPT P10636 1/20 0.37
RAB9A P51151 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2951931 0.78 PRKDC (0.42) DHFRXDHIGF1RCDK1CDK2
SCHEMBL2946044 0.76 MAPT (0.43) DHFRPOLBCDK1CDK2ATR
SCHEMBL2952943 0.75 MAP2K7 (0.45) PIK3CAPRKDC
SCHEMBL2946368 0.75 PRKDC (0.40) DHFRXDHCDK1CDK2MAPT
SCHEMBL2953061 0.69 DHFR (0.42) ADKDHFRPOLBCDK1CDK2
SCHEMBL24170032 0.68 AR (0.48) ADKJAK2JAK1TYK2JAK3
SCHEMBL521049 0.67 PIK3CA (0.56) ADKDHFRPOLBKDM4EMEN1
SCHEMBL29964578 0.66 PIK3CA (0.57) ADKXDHJAK2JAK1TYK2
SCHEMBL2558872 0.65 DHFR (0.60) ADKDHFRCDK1CDK2PIK3CA
SCHEMBL2949706 0.65 PIK3CA (0.57) DHFRPOLBKDM4EMAPTPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010111406-A2 COMPOUNDS AND THERAPEUTIC USES THEREOF MYRIAD PHARMACEUTICALS, INC. (US) 2010-09-30 WO claimed