SCHEMBL29535237

SCHEMBL29535237

COC(=O)c1ccc(Cl)c(NS(=O)(=O)c2ccc(C)cc2)c1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 5/20 0.76
LMNA P02545 6/20 0.68
HTT P42858 3/20 0.68
MAPT P10636 3/20 0.68
KDM4E B2RXH2 4/20 0.66
TSHR P16473 4/20 0.66
SMN1; SMN2 Q16637 1/20 0.66
ALDH1A1 P00352 9/20 0.63
NPSR1 Q6W5P4 1/20 0.62
TCF4 P15884 1/20 0.61
CTNNB1 P35222 1/20 0.61
HPGD P15428 1/20 0.55
CASP1 P29466 1/20 0.55
CASP7 P55210 1/20 0.55
HSD17B10 Q99714 1/20 0.55
FFAR4 Q5NUL3 1/20 0.54
PKM P14618 1/20 0.54
GAA P10253 1/20 0.53
MAPK1 P28482 1/20 0.52
FLT1 P17948 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16119560 1.00 CYP2C9 (0.76) CYP2C9LMNAHTTMAPTKDM4E
SCHEMBL7573928 0.88 CYP2C9 (0.82) CYP2C9LMNAHTTMAPTKDM4E
SCHEMBL21222732 0.86 LMNA (0.73) CYP2C9LMNAHTTMAPTKDM4E
SCHEMBL1073233 0.86 CYP2C9 (1.00) CYP2C9LMNAHTTMAPTKDM4E
SCHEMBL16318203 0.85 KDM4E (0.61) CYP2C9LMNAHTTMAPTKDM4E
SCHEMBL24102911 0.84 CYP2C9 (0.76) CYP2C9LMNAHTTMAPTKDM4E
SCHEMBL22391857 0.84 CYP2C9 (0.76) CYP2C9LMNAHTTMAPTKDM4E
SCHEMBL28560173 0.84 CYP2C9 (0.80) CYP2C9LMNAHTTKDM4ETSHR
SCHEMBL12787927 0.82 CYP2C9 (0.81) CYP2C9LMNAKDM4ETSHRSMN1; SMN2
SCHEMBL16438047 0.81 MAPT (0.64) CYP2C9LMNAHTTMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111285806-B Pyrazole compound and preparation method, application and pharmaceutical composition thereof 中国医学科学院药物研究所 2022-04-15 CN disclosed