SCHEMBL29548745

SCHEMBL29548745

CS(=O)(=O)Nc1cc(Br)c(Oc2ccc(F)cc2F)cc1C1CC1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.51
EPAS1 Q99814 1/20 0.45
BRD4 O60885 11/20 0.39
HTR1A P08908 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
HCRTR2 O43614 1/20 0.37
MAPK8 P45983 2/20 0.37
EP300 Q09472 1/20 0.37
MAPK14 Q16539 1/20 0.36
SCN9A Q15858 1/20 0.36
TRPV1 Q8NER1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28721123 1.00 PTGS2 (0.51) PTGS2EPAS1BRD4HTR1ASLC6A2
SCHEMBL29548605 0.89 BRD4 (0.46) PTGS2EPAS1BRD4MAPK14
SCHEMBL20443102 0.89 BRD4 (0.46) PTGS2EPAS1BRD4MAPK14
SCHEMBL16045757 0.85 PTGS2 (0.55) PTGS2EPAS1BRD4MAPK8EP300
SCHEMBL16045908 0.85 PTGS2 (0.61) PTGS2EPAS1BRD4MAPK8EP300
SCHEMBL16047515 0.81 PTGS2 (0.62) PTGS2EPAS1BRD4MAPK8EP300
SCHEMBL28721218 0.81 PTGS2 (0.48) PTGS2BRD4HTR1ASLC6A2SLC6A4
SCHEMBL29549380 0.81 PTGS2 (0.48) PTGS2BRD4HTR1ASLC6A2SLC6A4
SCHEMBL20443103 0.79 HTR1A (0.38) PTGS2EPAS1BRD4HTR1ASLC6A2
SCHEMBL29549365 0.79 PTGS2 (0.46) PTGS2BRD4EP300

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110041253-B Pyridine N-oxide derivative and preparation method and application thereof 上海翰森生物医药科技有限公司 2022-03-29 CN disclosed