SCHEMBL29548990

SCHEMBL29548990

NC(=O)c1cnc(-c2cccnc2)s1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.56
CYP2C19 P33261 2/20 0.56
CYP1A2 P05177 2/20 0.56
LMNA P02545 1/20 0.56
MKNK1 Q9BUB5 6/20 0.51
MKNK2 Q9HBH9 6/20 0.51
SMN1; SMN2 Q16637 2/20 0.49
NPC1 O15118 1/20 0.49
ALDH1A1 P00352 1/20 0.49
MAPT P10636 1/20 0.49
RAB9A P51151 1/20 0.49
GSK3B P49841 1/20 0.48
HPGDS O60760 1/20 0.48
CYP2A6 P11509 2/20 0.48
CYP2C9 P11712 1/20 0.48
KDM4E B2RXH2 1/20 0.47
CHEK1 O14757 1/20 0.47
HDAC1 Q13547 2/20 0.47
HDAC6 Q9UBN7 2/20 0.47
HDAC3 O15379 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5392323 1.00 CYP3A4 (0.56) CYP3A4CYP2C19CYP1A2LMNAMKNK1
SCHEMBL27768593 0.87 NPC1 (0.59) CYP3A4CYP2C19CYP1A2LMNAMKNK1
SCHEMBL1421843 0.86 MKNK1 (0.62) CYP3A4CYP2C19CYP1A2LMNAMKNK1
SCHEMBL14343335 0.84 CYP3A4 (0.63) CYP3A4CYP2C19CYP1A2LMNAMKNK1
SCHEMBL12725601 0.84 NPC1 (0.49) CYP3A4CYP2C19CYP1A2LMNAMKNK1
SCHEMBL892779 0.83 MAPT (0.68) CYP3A4CYP2C19CYP1A2SMN1; SMN2NPC1
Hydrochloric Acid SCHEMBL1421806 0.83 NPC1 (0.48) CYP3A4CYP2C19CYP1A2LMNAMKNK1
SCHEMBL10848656 0.82 CDC7 (0.61) CYP1A2SMN1; SMN2NPC1ALDH1A1MAPT
SCHEMBL11388698 0.82 ALDH1A1 (0.51) CYP3A4CYP2C19CYP1A2LMNAMKNK1
SCHEMBL24702452 0.81 HPGDS (0.54) CYP3A4CYP2C19CYP1A2LMNAMKNK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110167937-B Bicyclic bis-heteroaryl derivatives as modulators of protein aggregation UCB生物制药私人有限公司 2022-03-29 CN disclosed