SCHEMBL29575830

SCHEMBL29575830

CN1CCN(c2ccc(Nc3ncc4cccc(-c5ccncc5)c4n3)cc2)CC1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 2/20 0.66
BRD4 O60885 2/20 0.66
CDK4 P11802 7/20 0.58
AURKA O14965 4/20 0.58
CCND1 P24385 3/20 0.55
CCND2 P30279 3/20 0.55
CCND3 P30281 3/20 0.55
FGFR4 P22455 4/20 0.55
MAP4K1 Q92918 1/20 0.54
JAK3 P52333 1/20 0.54
JUN P05412 2/20 0.54
MAPK8 P45983 2/20 0.54
MAPK10 P53779 2/20 0.54
FGFR2 P21802 2/20 0.53
CCNB2 O95067 1/20 0.53
CCNE2 O96020 1/20 0.53
CDK1 P06493 1/20 0.53
FGFR1 P11362 1/20 0.53
CCNB1 P14635 1/20 0.53
CCNA2 P20248 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29576100 0.91 JAK2 (0.67) JAK2BRD4CDK4AURKACCND1
SCHEMBL18377046 0.87 BRD4 (0.63) JAK2BRD4CDK4AURKACCND1
SCHEMBL18376655 0.86 JAK2 (0.67) JAK2BRD4CDK4AURKACCND1
SCHEMBL1632115 0.85 JAK2 (0.66) JAK2BRD4CDK4AURKACCND1
SCHEMBL16514362 0.85 JAK2 (0.70) JAK2BRD4CDK4AURKACCND1
SCHEMBL29846917 0.85 JAK2 (0.70) JAK2BRD4CDK4AURKACCND1
SCHEMBL18377076 0.84 JAK2 (0.65) JAK2BRD4CDK4AURKACCND1
SCHEMBL28676614 0.84 JAK2 (0.61) JAK2BRD4CDK4AURKACCND1
SCHEMBL18376601 0.82 BRD4 (0.57) JAK2BRD4CDK4AURKACCND1
SCHEMBL18376804 0.81 JAK2 (0.57) JAK2BRD4CDK4AURKACCND1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260102406-A1 SUBSTITUTED QUINAZOLINES FOR INHIBITING KINASE ACTIVITY NEUPHARMA INC (US) 2026-04-16 US disclosed
US-12403145-B2 Substituted quinazolines for inhibiting kinase activity NEUPHARMA, INC (US) 2025-09-02 US disclosed
US-20240197752-A1 SUBSTITUTED QUINAZOLINES FOR INHIBITING KINASE ACTIVITY NEUPHARMA INC 2024-06-20 US disclosed
US-11865120-B2 Substituted quinazolines for inhibiting kinase activity NEUPHARMA, INC. (US) 2024-01-09 US disclosed
US-20220354864-A1 SUBSTITUTED QUINAZOLINES FOR INHIBITING KINASE ACTIVITY NEUPHARMA, INC. 2022-11-10 US disclosed
US-11304957-B2 Substituted quinazolines for inhibiting kinase activity NEUPHARMA, INC. (US) 2022-04-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240197752-A1 SUBSTITUTED QUINAZOLINES FOR INHIBITING KINASE ACTIVITY DCK, ABL1, MAP4K2 JAK2 356/4885BRD4 474/4885CDK4 156/4885
US-11865120-B2 Substituted quinazolines for inhibiting kinase activity DCK, ABL1, MAP4K2 JAK2 356/4885BRD4 474/4885CDK4 156/4885
US-12403145-B2 Substituted quinazolines for inhibiting kinase activity DCK, ABL1, MAP4K2 JAK2 356/4885BRD4 474/4885CDK4 156/4885
US-11304957-B2 Substituted quinazolines for inhibiting kinase activity DCK, ABL1, MAP4K2 JAK2 356/4885BRD4 474/4885CDK4 156/4885
US-20220354864-A1 SUBSTITUTED QUINAZOLINES FOR INHIBITING KINASE ACTIVITY DCK, ABL1, MAP4K2 JAK2 356/4885BRD4 474/4885CDK4 156/4885
US-20260102406-A1 SUBSTITUTED QUINAZOLINES FOR INHIBITING KINASE ACTIVITY BRAF, TTK, MAP4K2 JAK2 155/4885BRD4 1922/4885CDK4 358/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.