SCHEMBL29581998

SCHEMBL29581998

CCOC(=O)c1cnc(SCc2ccc([N+](=O)[O-])c(C(F)(F)F)c2)[nH]c1=O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 4/20 0.47
CA1 P00915 4/20 0.47
CA2 P00918 4/20 0.47
CA6 P23280 4/20 0.47
CA7 P43166 4/20 0.47
CA13 Q8N1Q1 4/20 0.47
KDM4E B2RXH2 4/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
KDM6B O15054 1/20 0.41
KDM4A O75164 1/20 0.41
KDM4D Q6B0I6 1/20 0.41
HIF1AN Q9NWT6 1/20 0.41
KDM5B Q9UGL1 1/20 0.41
KDM2A Q9Y2K7 1/20 0.41
DAO P14920 2/20 0.41
GSTP1 P09211 1/20 0.41
GSTM2 P28161 1/20 0.41
ALDH1A1 P00352 3/20 0.40
GAA P10253 1/20 0.40
MEN1 O00255 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29581252 0.86 KDM6B (0.45) KDM6BKDM4AKDM4DHIF1ANKDM5B
SCHEMBL3583829 0.78 KDM6B (0.55) CA12CA1CA2CA6CA7
SCHEMBL9900826 0.78 CA12 (0.49) CA12CA1CA2CA6CA7
SCHEMBL22867798 0.78 CA12 (0.50) CA12CA1CA2CA6CA7
SCHEMBL29581389 0.78 CA12 (0.50) CA12CA1CA2CA6CA7
SCHEMBL29581651 0.74 HSD17B2 (0.51) DAO
SCHEMBL22868062 0.71 CA12 (0.47) CA12CA1CA2CA6CA7
SCHEMBL6593772 0.70 AR (0.56) CA12L3MBTL1ALDH1A1LMNAMAPT
SCHEMBL11013238 0.69 CA12 (0.57) CA12CA1CA2CA6CA7
SCHEMBL3160169 0.68 KDM6B (0.63) CA12CA1CA2CA6CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3994125-A1 MODULATORS OF HSD17B13 AND METHODS OF USE THEREOF Regeneron Pharmaceuticals, Inc. (US) 2022-05-11 EP disclosed