SCHEMBL29586304

SCHEMBL29586304

OB(O)c1ccc(N2CCOCC2)nc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.54
CNR2 P34972 8/20 0.51
HPGD P15428 3/20 0.51
HSD17B10 Q99714 3/20 0.51
MAPT P10636 3/20 0.51
KDM4E B2RXH2 2/20 0.51
CYP1A2 P05177 2/20 0.51
LMNA P02545 2/20 0.51
HTT P42858 2/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
CYP2C9 P11712 1/20 0.51
MEN1 O00255 1/20 0.51
GAA P10253 1/20 0.51
RECQL P46063 1/20 0.51
KMT2A Q03164 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
POLB P06746 1/20 0.50
ALOX15 P16050 1/20 0.50
AKR1C3 P42330 1/20 0.47
CYP2C19 P33261 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9147 1.00 ALDH1A1 (0.54) ALDH1A1CNR2HPGDHSD17B10MAPT
SCHEMBL14167546 0.94 CNR2 (0.53) ALDH1A1CNR2HPGDHSD17B10MAPT
SCHEMBL28629103 0.91 ALDH1A1 (0.48) ALDH1A1CNR2HPGDHSD17B10MAPT
SCHEMBL29377204 0.84 UBE2T (0.51) ALDH1A1CNR2HPGDHSD17B10MAPT
SCHEMBL676085 0.84 UBE2T (0.51) ALDH1A1CNR2HPGDHSD17B10MAPT
SCHEMBL3941056 0.83 UBE2T (0.50) ALDH1A1CNR2HPGDHSD17B10MAPT
SCHEMBL29951531 0.83 UBE2T (0.50) ALDH1A1CNR2HPGDHSD17B10MAPT
SCHEMBL29951844 0.83 UBE2T (0.50) ALDH1A1CNR2HPGDHSD17B10MAPT
SCHEMBL2562848 0.80 HTR3A (0.47) ALDH1A1KDM4ECYP1A2SMN1; SMN2KMT2A
SCHEMBL723901 0.80 PLD1 (0.49) ALDH1A1HPGDHSD17B10KDM4ECYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232090-A 6-substituted dihydrobenzo [ e ] [1,2,3] oxathiazine 2,2-dioxide compound and preparation and application thereof 杭州市第七人民医院 2022-10-25 CN claimed
CN-116162087-B HPK 1 and/or LCK kinase regulator, preparation method and application thereof 杭州医学院 2024-07-23 CN disclosed
EP-4313967-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2024-02-07 EP disclosed
EP-4255906-A1 NEW INDAZOLE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2023-10-11 EP disclosed
CN-115232090-A 6-substituted dihydrobenzo [ e ] [1,2,3] oxathiazine 2,2-dioxide compound and preparation and application thereof 杭州市第七人民医院 2022-10-25 CN disclosed
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed
WO-2022117487-A1 NEW INDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2022-06-09 WO disclosed