SCHEMBL29587246

SCHEMBL29587246

O=C(NO)C1CCc2ccc(OCc3ccc(Cl)cc3)cc2O1

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAOB P27338 6/20 0.48
CYP4F2 P78329 2/20 0.48
CYP4A11 Q02928 2/20 0.48
HTR6 P50406 1/20 0.46
MAOA P21397 5/20 0.45
ADAM17 P78536 2/20 0.45
PPARG P37231 2/20 0.44
PPARD Q03181 2/20 0.44
PPARA Q07869 2/20 0.44
MMP1 P03956 1/20 0.43
SMPD1 P17405 1/20 0.43
ITGB3 P05106 1/20 0.43
ITGA2B P08514 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29586744 0.89 NPC1 (0.49) MAOBCYP4F2CYP4A11HTR6MAOA
SCHEMBL29588068 0.89 MAOB (0.48) MAOBCYP4F2CYP4A11HTR6MAOA
SCHEMBL29587734 0.88 CYP4F2 (0.59) MAOBCYP4F2CYP4A11HTR6MAOA
SCHEMBL27091892 0.87 MAOB (0.47) MAOBCYP4F2CYP4A11HTR6MAOA
SCHEMBL29588124 0.83 ADAM17 (0.46) MAOBCYP4F2CYP4A11HTR6MAOA
SCHEMBL29587114 0.83 CYP4F2 (0.56) MAOBCYP4F2CYP4A11HTR6MAOA
SCHEMBL29586899 0.82 MAOB (0.43) MAOBCYP4F2CYP4A11HTR6MAOA
SCHEMBL29586818 0.82 ADAM17 (0.52) MAOBCYP4F2CYP4A11HTR6ADAM17
SCHEMBL29588229 0.79 PPARG (0.51) MAOBCYP4F2CYP4A11HTR6MAOA
SCHEMBL27091891 0.78 PPARG (0.48) MAOBCYP4F2CYP4A11MAOAPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022120048-A1 HDAC INHIBITORS UNIVERSITY OF PITTSBURGH - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2022-06-09 WO disclosed