SCHEMBL29595384

SCHEMBL29595384

CSc1ncc(CO)c(N[C@@H]2COCC2(C)O)n1

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.39
NR3C1 P04150 1/20 0.37
PGR P06401 1/20 0.37
AR P10275 1/20 0.37
MERTK Q12866 1/20 0.31
TYK2 P29597 2/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19863579 1.00 HTT (0.39) HTTNR3C1PGRARMERTK
SCHEMBL29798910 1.00 HTT (0.39) HTTNR3C1PGRARMERTK
SCHEMBL19857322 0.81 HTT (0.40) HTTNR3C1PGRARMERTK
SCHEMBL29507789 0.81 HTT (0.40) HTTNR3C1PGRARMERTK
SCHEMBL29594214 0.81 HTT (0.40) HTTNR3C1PGRARMERTK
SCHEMBL19857380 0.81 HTT (0.40) HTTNR3C1PGRARMERTK
SCHEMBL20955932 0.81 NR3C1 (0.36) NR3C1PGRARTYK2ALDH1A1
SCHEMBL20955933 0.81 NR3C1 (0.36) NR3C1PGRARTYK2ALDH1A1
SCHEMBL19863577 0.78 ALDH1A1 (0.53) HTTALDH1A1MAPTSMN1; SMN2
SCHEMBL20955940 0.77 HTT (0.39) HTTMERTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114394966-A Pyridopyrimidinone CDK2/4/6 inhibitors 辉瑞公司 2022-04-26 CN disclosed