SCHEMBL29601607

SCHEMBL29601607

Cc1cccnc1C(=O)NCC(=O)O

nearest known ligand 0.69

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
FTO Q9C0B1 2/20 0.69
EGLN2 Q96KS0 1/20 0.69
EGLN1 Q9GZT9 14/20 0.51
GAA P10253 1/20 0.51
VEGFA P15692 2/20 0.47
FLT1 P17948 2/20 0.47
EGLN3 Q9H6Z9 1/20 0.47
ITGB3 P05106 1/20 0.46
ITGB1 P05556 1/20 0.46
ITGAV P06756 1/20 0.46
ITGA5 P08648 1/20 0.46
KDM5B Q9UGL1 1/20 0.46
KDM2A Q9Y2K7 1/20 0.46
CTSA P10619 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27039728 1.00 FTO (0.69) FTOEGLN2EGLN1GAAVEGFA
SCHEMBL10709742 0.84 EGLN2 (0.49) FTOEGLN2CTSA
SCHEMBL13310736 0.83 PARP1 (0.48) FTOEGLN2
SCHEMBL704958 0.82 FTO (1.00) FTOEGLN2EGLN1VEGFAFLT1
SCHEMBL29601361 0.82 ALDH1A1 (0.51) FTOEGLN2
SCHEMBL3958929 0.81 KMT2A (0.61) EGLN1GAA
SCHEMBL8883374 0.81 FTO (0.69) FTOEGLN2EGLN1GAAKDM5B
SCHEMBL22804019 0.81 FTO (0.69) FTOEGLN2EGLN1GAAKDM5B
SCHEMBL704947 0.80 EGLN2 (0.64) FTOEGLN2EGLN1GAACTSA
SCHEMBL109198 0.80 P2RX7 (0.59) FTOEGLN2GAACTSA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4232449-A1 HETEROCYCLIC COMPOUNDS AND THEIR USE FOR TREATMENT OF HELMINTHIC INFECTIONS AND DISEASES Celgene Corporation (US) 2023-08-30 EP disclosed
WO-2022087326-A1 HETEROCYCLIC COMPOUNDS AND THEIR USE FOR TREATMENT OF HELMINTHIC INFECTIONS AND DISEASES CELGENE CORPORATION (US) 2022-04-28 WO disclosed