SCHEMBL29604688

SCHEMBL29604688

O=C1N(CC(F)(F)F)CC[C@@]1(O)c1cccc(Br)c1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 2/20 0.33
P2RX7 Q99572 1/20 0.33
CHRNA1 P02708 1/20 0.33
CHRNG P07510 1/20 0.33
CHRNB1 P11230 1/20 0.33
CHRNB2 P17787 1/20 0.33
SLC6A2 P23975 1/20 0.33
CHRNB4 P30926 1/20 0.33
SLC6A4 P31645 1/20 0.33
CHRNA3 P32297 1/20 0.33
CHRNA4 P43681 1/20 0.33
SLC6A3 Q01959 1/20 0.33
CHRND Q07001 1/20 0.33
OPRM1 P35372 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
OPRD1 P41143 1/20 0.33
OPRK1 P41145 1/20 0.33
ALDH1A1 P00352 3/20 0.32
TP53 P04637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29604773 1.00 HSD11B1 (0.33) HSD11B1P2RX7CHRNA1CHRNGCHRNB1
SCHEMBL26969531 1.00 HSD11B1 (0.33) HSD11B1P2RX7CHRNA1CHRNGCHRNB1
SCHEMBL26969399 0.80 LIPG (0.35) OPRM1OPRD1OPRK1
SCHEMBL27121386 0.80 LIPG (0.35) OPRM1OPRD1OPRK1
SCHEMBL29604635 0.80 LIPG (0.35) OPRM1OPRD1OPRK1
SCHEMBL29604777 0.76 GRIN1 (0.43) HSD11B1CHRNA1CHRNGCHRNB1CHRNB2
SCHEMBL26644185 0.76 GRIN1 (0.43) HSD11B1CHRNA1CHRNGCHRNB1CHRNB2
SCHEMBL29604803 0.76 GRIN1 (0.43) HSD11B1CHRNA1CHRNGCHRNB1CHRNB2
SCHEMBL26644188 0.76 GRIN1 (0.43) HSD11B1CHRNA1CHRNGCHRNB1CHRNB2
SCHEMBL29604868 0.71 GRIN1 (0.47) HSD11B1CHRNA1CHRNGCHRNB1CHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4244224-A1 SMALL MOLECULE INHIBITORS OF NF-KB INDUCING KINASE JANSSEN Pharmaceutica NV (BE) 2023-09-20 EP disclosed
WO-2022104348-A1 SMALL MOLECULE INHIBITORS OF NF-KB INDUCING KINASE JANSSEN PHARMACEUTICA NV (BE) 2022-05-19 WO disclosed