SCHEMBL29612142

SCHEMBL29612142

C[C@H]1Cc2sc3ccccc3c2[C@H](c2ccc(I)cc2)N1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PNMT P11086 1/20 0.33
CYP1A1 P04798 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30
HTR2A P28223 1/20 0.30
CYP2C19 P33261 1/20 0.30
GPR3 P46089 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19760754 1.00 PNMT (0.33) PNMTCYP1A1CYP1A2CYP3A4CYP2D6
SCHEMBL19760752 1.00 PNMT (0.33) PNMTCYP1A1CYP1A2CYP3A4CYP2D6
SCHEMBL24026964 0.88 CCKBR (0.35) PNMTCYP1A1CYP1A2CYP3A4CYP2D6
SCHEMBL29317134 0.67 GPR3 (0.40) PNMTCYP1A1CYP1A2CYP3A4CYP2D6
SCHEMBL3062843 0.67 GRIN2D (0.42)
SCHEMBL19760715 0.66 GPER1 (0.37) PNMT
SCHEMBL29611854 0.64 PNMT (0.62) PNMT
SCHEMBL26837118 0.63 PNMT (0.50) PNMT
SCHEMBL24026979 0.60 GPER1 (0.38) PNMT
SCHEMBL30071485 0.57 GPR3 (0.35) PNMTGPR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109311876-B Heteroaryl estrogen receptor modulators and uses thereof 豪夫迈·罗氏有限公司 2022-05-03 CN disclosed