SCHEMBL29615396

SCHEMBL29615396

COc1ncc(C#N)cc1-c1ccc(C(F)(F)F)cn1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 2/20 0.41
KDM1A O60341 2/20 0.39
KDM4E B2RXH2 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
HPGDS O60760 2/20 0.37
GRM5 P41594 2/20 0.37
MAOB P27338 2/20 0.37
TRPV1 Q8NER1 1/20 0.37
ALDH1A1 P00352 1/20 0.36
TSHR P16473 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
PGR P06401 1/20 0.36
PTGDR2 Q9Y5Y4 2/20 0.36
KIF11 P52732 1/20 0.36
PDE1B Q01064 1/20 0.35
PDE1C Q14123 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20577824 1.00 NR3C1 (0.41) NR3C1KDM1AKDM4ENPSR1HPGDS
SCHEMBL29615607 0.84 NR3C1 (0.51) NR3C1KDM1AHPGDSMAOBPGR
SCHEMBL20577702 0.84 NR3C1 (0.51) NR3C1KDM1AHPGDSMAOBPGR
SCHEMBL18223690 0.82 KDM1A (0.58) KDM1AALDH1A1TSHRSMN1; SMN2PTGDR2
SCHEMBL20577865 0.77 SCN9A (0.39) KDM1AKDM4ENPSR1ALDH1A1TSHR
SCHEMBL29615348 0.77 SCN9A (0.39) KDM1AKDM4ENPSR1ALDH1A1TSHR
SCHEMBL18002768 0.74 GRM5 (0.59) KDM1AKDM4ENPSR1GRM5SMN1; SMN2
SCHEMBL2707348 0.73 LRRK2 (0.43) NR3C1KDM4EHPGDSPGRKIF11
SCHEMBL18223968 0.71 CYP1A2 (0.48) KDM4ENPSR1GRM5MAOBTRPV1
SCHEMBL10460598 0.70 CYP1A2 (0.40) KDM4EALDH1A1PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108602807-B Heterocyclic sulfonamide derivatives and drugs containing the same EA制药株式会社 2022-05-13 CN disclosed