SCHEMBL29616448

SCHEMBL29616448

FC(F)(F)c1ccc(CBr)cc1-c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 2/20 0.40
PTPN1 P18031 1/20 0.40
KIF11 P52732 1/20 0.39
TRPA1 O75762 1/20 0.39
ALDH1A1 P00352 1/20 0.39
TSHR P16473 1/20 0.39
TACR1 P25103 3/20 0.38
SLC13A5 Q86YT5 1/20 0.38
RXRA P19793 1/20 0.37
RXRB P28702 1/20 0.37
RXRG P48443 1/20 0.37
HSD11B1 P28845 1/20 0.36
USP1 O94782 1/20 0.36
WDR48 Q8TAF3 1/20 0.36
BACE1 P56817 1/20 0.36
PDCD1 Q15116 2/20 0.36
CD274 Q9NZQ7 2/20 0.36
PSEN1 P49768 1/20 0.36
PSEN2 P49810 1/20 0.36
APH1B Q8WW43 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23148953 1.00 CNR2 (0.40) CNR2PTPN1KIF11TRPA1ALDH1A1
SCHEMBL2324650 0.84 KIF11 (0.51) CNR2PTPN1KIF11TSHRSLC13A5
SCHEMBL5726820 0.79 SLC13A5 (0.49) CNR2TRPA1ALDH1A1TSHRSLC13A5
SCHEMBL1373277 0.77 ALDH1A1 (0.48) PTPN1TRPA1ALDH1A1TSHRBACE1
SCHEMBL5050345 0.76 PSEN1 (0.47) ALDH1A1TACR1SLC13A5PSEN1PSEN2
SCHEMBL4663038 0.75 MAOB (0.41)
SCHEMBL1775215 0.75 RXRA (0.44) KIF11TRPA1ALDH1A1TSHRRXRA
SCHEMBL2300881 0.74 KIF11 (0.54) KIF11ALDH1A1TSHRTACR1BACE1
SCHEMBL3764165 0.74 ALDH1A1 (0.44) PTPN1TRPA1ALDH1A1TSHRTACR1
SCHEMBL15075513 0.74 ALDH1A1 (0.50) PTPN1TRPA1ALDH1A1TSHRBACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114401968-A Novel heterocyclic monoacylglycerol lipase (MAGL) inhibitors 豪夫迈·罗氏有限公司 2022-04-26 CN disclosed