SCHEMBL29618364

SCHEMBL29618364

O=C1OC(O)(C(F)(F)F)c2cc(Br)ccc21

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 5/20 0.53
OPRM1 P35372 1/20 0.44
OPRD1 P41143 1/20 0.44
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA4 P22748 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
AKR1C1 Q04828 1/20 0.36
S100A4 P26447 1/20 0.35
PTPRC P08575 1/20 0.35
AKR1A1 P14550 1/20 0.35
AKR1B1 P15121 1/20 0.35
BCL2 P10415 1/20 0.34
MCL1 Q07820 1/20 0.34
TDP2 O95551 1/20 0.34
HSP90AA1 P07900 1/20 0.34
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24517455 1.00 PDK2 (0.53) PDK2OPRM1OPRD1CA1CA2
SCHEMBL29618362 1.00 PDK2 (0.53) PDK2OPRM1OPRD1CA1CA2
SCHEMBL28758440 0.89 PDK2 (0.46) PDK2OPRM1OPRD1CA1CA2
SCHEMBL31202620 0.80 PDK2 (0.53) PDK2AKR1C1HSP90AA1ALDH1A1MAPT
SCHEMBL10554281 0.80 PDK2 (0.53) PDK2AKR1C1HSP90AA1ALDH1A1MAPT
SCHEMBL31073015 0.76 OPRM1 (0.47) PDK2OPRM1OPRD1CA1CA2
SCHEMBL23526283 0.75 PDK2 (0.42) PDK2OPRM1OPRD1CA1CA2
SCHEMBL16064982 0.71 OPRM1 (0.46) PDK2OPRM1OPRD1CA1CA2
SCHEMBL29922211 0.71 OPRM1 (0.46) PDK2OPRM1OPRD1CA1CA2
SCHEMBL12460624 0.69 PDK2 (1.00) PDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114591293-A Fused ring compound as Nav1.8 inhibitor and application thereof 成都康弘药业集团股份有限公司 2022-06-07 CN disclosed