SCHEMBL29633677

SCHEMBL29633677

Cc1cccc(CC(NC(=O)OCC2c3ccccc3-c3ccccc32)C(=O)OC(C)(C)C)c1

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MDM4 O15151 1/20 0.46
TP53 P04637 1/20 0.46
MAPT P10636 1/20 0.45
NTSR1 P30989 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
POLB P06746 1/20 0.44
EPHX2 P34913 1/20 0.43
PTPN1 P18031 2/20 0.43
MDM2 Q00987 1/20 0.43
CTSB P07858 1/20 0.43
CTSS P25774 1/20 0.43
CTSK P43235 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28741469 0.90 MDM4 (0.45) MDM4TP53EPHX2MDM2CTSS
SCHEMBL29634043 0.90 MDM4 (0.45) MDM4TP53EPHX2MDM2CTSS
SCHEMBL28741504 0.90 MDM4 (0.52) MDM4TP53MAPTTDP1POLB
SCHEMBL28741502 0.90 MDM4 (0.52) MDM4TP53MAPTTDP1POLB
SCHEMBL28741567 0.89 CTSL (0.52) MDM4TP53MAPTNPSR1EPHX2
SCHEMBL29633851 0.89 MDM2 (0.48) MDM4TP53PTPN1MDM2
SCHEMBL28741521 0.89 MDM4 (0.45) MDM4TP53EPHX2PTPN1MDM2
SCHEMBL22454530 0.89 MDM4 (0.47) MDM4TP53POLBPTPN1MDM2
SCHEMBL16095370 0.88 MDM4 (0.52) MDM4TP53POLBEPHX2PTPN1
SCHEMBL30343679 0.88 MDM4 (0.52) MDM4TP53POLBEPHX2PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240376044-A1 METHOD FOR PREPARING AROMATIC AMINO ACID DERIVATIVE CHUGAI PHARMACEUTICAL CO LTD (JP) 2024-11-14 US disclosed
US-12071396-B2 Method for preparing aromatic amino acid derivative CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2024-08-27 US disclosed
US-20220144762-A1 METHOD FOR PREPARING AROMATIC AMINO ACID DERIVATIVE CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2022-05-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240376044-A1 METHOD FOR PREPARING AROMATIC AMINO ACID DERIVATIVE DDC, AADAT, TYR MDM4 381/4885TP53 1369/4885MAPT 1196/4885
US-20220144762-A1 METHOD FOR PREPARING AROMATIC AMINO ACID DERIVATIVE DDC, AADAT, TYR MDM4 381/4885TP53 1369/4885MAPT 1196/4885
US-12071396-B2 Method for preparing aromatic amino acid derivative DDC, AADAT, TYR MDM4 381/4885TP53 1369/4885MAPT 1196/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.