Betazole

Betazole

SCHEMBL29633745

Cl.Cl.NCCc1ccn[nH]1

nearest known ligand 0.95

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

HRH2

The experimentally established mechanism targets of Betazole. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HRH2 known ✓ P25021 3/20 0.95
USP2 O75604 2/20 0.95
LMNA P02545 2/20 0.95
HRH4 Q9H3N8 3/20 0.42
HRH3 Q9Y5N1 2/20 0.42
APEX1 P27695 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
TSHR P16473 2/20 0.39
HRH1 P35367 5/20 0.39
MIF P14174 1/20 0.39
LOXL2 Q9Y4K0 1/20 0.38
AKT2 P31751 1/20 0.33
CHRNA7 P36544 1/20 0.33
KCNH2 Q12809 1/20 0.33
HTR1B P28222 1/20 0.33
BLM P54132 1/20 0.32
KMT2A Q03164 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
KDM4C Q9H3R0 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Betazole SCHEMBL1237745 1.00
Betazole SCHEMBL3336050 0.98 HRH2 (1.00) HRH2USP2LMNAHRH4HRH3
Betazole SCHEMBL157156 0.98
Betazole SCHEMBL1649674 0.95 HRH2 (0.95) HRH2USP2LMNAHRH4HRH3
SCHEMBL4711257 0.84
Betazole SCHEMBL3336046 0.80 USP2 (0.68) HRH2USP2LMNAHRH4HRH3
SCHEMBL2183872 0.78
SCHEMBL21721708 0.74
SCHEMBL4222977 0.74
Bromide SCHEMBL10400923 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 40 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117996825-A Optimal control method for cogeneration based on hydrogen fuel cell technology 国网山东省电力公司电力科学研究院 2024-05-07 CN claimed
EP-4251163-A1 ANTI-VIRAL ACTIVITY OF VPS34 INHIBITORS Deciphera Pharmaceuticals, LLC (US) 2023-10-04 EP claimed
EP-4251167-A1 ANTI-VIRAL ACTIVITY OF VPS34 INHIBITORS Deciphera Pharmaceuticals, LLC (US) 2023-10-04 EP claimed
EP-4251165-A1 MORPHOLINO DERIVATIVES AS VSP34 INHIBITORS FOR USE IN THE TREATMENT OF A VIRAL INFECTION Deciphera Pharmaceuticals, LLC (US) 2023-10-04 EP claimed
EP-4251152-A1 PYRIDYLPYRIDONE DERIVATIVES AS VSP34 INHIBITORS FOR USE IN THE TREATMENT OF A VIRAL INFECTION Deciphera Pharmaceuticals, LLC (US) 2023-10-04 EP claimed
EP-4251156-A1 ANTI-VIRAL ACTIVITY OF VPS34 INHIBITORS Deciphera Pharmaceuticals, LLC (US) 2023-10-04 EP claimed
WO-2022115546-A1 ANTI-VIRAL ACTIVITY OF VPS34 INHIBITORS DECIPHERA PHARMACEUTICALS, LLC (US) 2022-06-02 WO claimed
WO-2022115545-A1 PYRIDYLPYRIDONE DERIVATIVES AS VSP34 INHIBITORS FOR USE IN THE TREATMENT OF A VIRAL INFECTION DECIPHERA PHARMACEUTICALS, LLC (US) 2022-06-02 WO claimed
WO-2022115558-A1 MORPHOLINO DERIVATIVES AS VSP34 INHIBITORS FOR USE IN THE TREATMENT OF A VIRAL INFECTION DECIPHERA PHARMACEUTICALS, LLC (US) 2022-06-02 WO claimed
WO-2022115549-A1 ANTI-VIRAL ACTIVITY OF VPS34 INHIBITORS DECIPHERA PHARMACEUTICALS, LLC (US) 2022-06-02 WO claimed
WO-2022115543-A1 ANTI-VIRAL ACTIVITY OF VPS34 INHIBITORS DECIPHERA PHARMACEUTICALS, LLC (US) 2022-06-02 WO claimed
WO-2026043901-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS OF TREATING ENTEROVIRUSES WITH VAPENDAVIR SULFATE Altesa BioSciences, Inc. (US) 2026-02-26 WO disclosed
US-20260048050-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS OF TREATING ENTEROVIRUSES WITH VAPENDAVIR SULFATE Altesa BioSciences, Inc. (US) 2026-02-19 US disclosed
US-12453717-B1 Methods of treating symptoms of coronavirus infection with viral protease inhibitors Accencio LC (US) 2025-10-28 US disclosed
US-12414955-B2 Anti-viral activity of VPS34 inhibitors DECIPHERA PHARMACEUTICALS, LLC (US) 2025-09-16 US disclosed
WO-2022115543-A1 ANTI-VIRAL ACTIVITY OF VPS34 INHIBITORS DECIPHERA PHARMACEUTICALS, LLC (US) 2022-06-02 WO disclosed
WO-2022115546-A1 ANTI-VIRAL ACTIVITY OF VPS34 INHIBITORS DECIPHERA PHARMACEUTICALS, LLC (US) 2022-06-02 WO disclosed
WO-2022115558-A1 MORPHOLINO DERIVATIVES AS VSP34 INHIBITORS FOR USE IN THE TREATMENT OF A VIRAL INFECTION DECIPHERA PHARMACEUTICALS, LLC (US) 2022-06-02 WO disclosed
WO-2022115545-A1 PYRIDYLPYRIDONE DERIVATIVES AS VSP34 INHIBITORS FOR USE IN THE TREATMENT OF A VIRAL INFECTION DECIPHERA PHARMACEUTICALS, LLC (US) 2022-06-02 WO disclosed
WO-2022115549-A1 ANTI-VIRAL ACTIVITY OF VPS34 INHIBITORS DECIPHERA PHARMACEUTICALS, LLC (US) 2022-06-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12414955-B2 Anti-viral activity of VPS34 inhibitors SARS1, VPS26B, VPS4B HRH2 4366/4885USP2 249/4885LMNA 3975/4885
US-12453717-B1 Methods of treating symptoms of coronavirus infection with viral protease inhibitors ACE, ACE2, TMPRSS2 HRH2 3545/4885USP2 796/4885LMNA 2391/4885
US-20260048050-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS OF TREATING ENTEROVIRUSES WITH VAPENDAVIR SULFATE RPP30, EXOSC9, RPL30 HRH2 1570/4885USP2 4260/4885LMNA 3746/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.