SCHEMBL29636159

SCHEMBL29636159

Cc1cnc(CCl)c(F)c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.34
CCR5 P51681 1/20 0.34
CCR8 P51685 1/20 0.34
NOS3 P29474 1/20 0.34
NOS1 P29475 1/20 0.34
NOS2 P35228 1/20 0.34
AGBL2 Q5U5Z8 1/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2B Q13224 1/20 0.33
CHRM2 P08172 1/20 0.33
CHRM4 P08173 1/20 0.33
CHRM5 P08912 1/20 0.33
CHRM1 P11229 1/20 0.33
CHRM3 P20309 1/20 0.33
CXCR4 P61073 1/20 0.33
KDM4E B2RXH2 1/20 0.32
CYP1A2 P05177 1/20 0.31
P2RX3 P56373 1/20 0.31
P2RX2 Q9UBL9 1/20 0.31
ALOX5AP P20292 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16039165 1.00 CCR1 (0.34) CCR1CCR5CCR8NOS3NOS1
SCHEMBL30854431 0.84 CCR1 (0.32) CCR1CCR5CCR8NOS3NOS1
SCHEMBL20261166 0.83 CCR1 (0.37) CCR1CCR5CCR8NOS3NOS1
SCHEMBL4132951 0.81 NOS3 (0.35) CCR1CCR5CCR8NOS3NOS1
SCHEMBL13732029 0.79 NOS3 (0.39) CCR1CCR5CCR8NOS3NOS1
SCHEMBL16741027 0.79 AGBL2 (0.37) CCR1CCR5CCR8NOS3NOS1
SCHEMBL26971130 0.79 CHRM2 (0.35) CCR1CCR5CCR8NOS3NOS1
SCHEMBL30164264 0.78 NOS3 (0.46) CCR1CCR5CCR8NOS3NOS1
SCHEMBL286660 0.78 NOS3 (0.46) CCR1CCR5CCR8NOS3NOS1
SCHEMBL29475252 0.78 AGBL2 (0.39) AGBL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119176794-A Heterocyclic compound, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2024-12-24 CN disclosed
CN-114989164-B Substituted 1H-imidazo [4,5-b ] pyridin-2 (3H) -ones and uses thereof 詹森药业有限公司 2024-08-13 CN disclosed
CN-114989164-A Substituted 1H-imidazo [4,5-b ] pyridin-2 (3H) -ones and uses thereof 詹森药业有限公司 2022-09-02 CN disclosed
CN-110062761-B Substituted 1H-imidazo [4,5-b ] pyridin-2 (3H) -ones and uses thereof 詹森药业有限公司 2022-05-13 CN disclosed