SCHEMBL29636347

SCHEMBL29636347

C=C(C)c1nc(N)c2cccn2n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 1/20 0.41
LMNA P02545 1/20 0.36
EGFR P00533 1/20 0.36
SPR P35270 2/20 0.33
PAX8 Q06710 1/20 0.32
MEN1 O00255 1/20 0.31
PDE5A O76074 1/20 0.31
ALDH1A1 P00352 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
MIF P14174 1/20 0.31
TSHR P16473 1/20 0.31
PDE4A P27815 1/20 0.31
ADORA2A P29274 1/20 0.31
ADORA1 P30542 1/20 0.31
CYP2C19 P33261 1/20 0.31
BLM P54132 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5080208 0.74 MAP4K4 (0.47) MAP4K4EGFRALDH1A1ADORA2AADORA1
SCHEMBL807452 0.73 MAP4K4 (0.50) MAP4K4EGFRPIK3CDPIK3R1PIK3CA
SCHEMBL807453 0.70 MAP4K4 (0.47) MAP4K4EGFRADORA2AADORA1PIK3CD
SCHEMBL30989127 0.70 MAP4K4 (0.47) MAP4K4EGFRADORA2APIK3CDPIK3R1
SCHEMBL12314541 0.70 MAP4K4 (0.47) MAP4K4LMNAEGFRPDE5AALDH1A1
SCHEMBL29350296 0.70 MAP4K4 (0.47) MAP4K4EGFRPIK3CDPIK3R1PIK3CA
SCHEMBL25273564 0.68 MAP4K4 (0.41) MAP4K4EGFRMEN1PDE5AALDH1A1
SCHEMBL30280494 0.68 MAP4K4 (0.41) MAP4K4LMNAEGFRCYP1A2CYP2D6
SCHEMBL25270993 0.68 BAZ1A (0.41) LMNAMEN1ALDH1A1CYP3A4CYP2D6
SCHEMBL16635772 0.67 MAP4K4 (0.40) MAP4K4EGFRPIK3CDPIK3R1PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114621233-A Substituted aromatic condensed ring derivative and its composition and use 深圳市塔吉瑞生物医药有限公司 2022-06-14 CN disclosed
CN-112552302-B Substituted aromatic fused ring derivatives, compositions and uses thereof 深圳市塔吉瑞生物医药有限公司 2022-05-13 CN disclosed