SCHEMBL29636830

SCHEMBL29636830

CC(=O)Nc1ccc(-c2nc3ccccc3s2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 7/20 0.74
KDM4E B2RXH2 6/20 0.74
NPC1 O15118 5/20 0.74
SMN1; SMN2 Q16637 5/20 0.74
TP53 P04637 4/20 0.74
GAA P10253 3/20 0.74
MMP2 P08253 1/20 0.71
MMP9 P14780 1/20 0.71
MMP8 P22894 1/20 0.71
MMP13 P45452 1/20 0.71
SULT1A1 P50225 1/20 0.70
MAPT P10636 4/20 0.67
MEN1 O00255 5/20 0.67
KMT2A Q03164 5/20 0.67
APP P05067 1/20 0.67
GLA P06280 1/20 0.67
MGLL Q99685 5/20 0.65
ALDH1A1 P00352 3/20 0.62
POLB P06746 2/20 0.62
PKM P14618 2/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7105704 1.00 RAB9A (0.74) RAB9AKDM4ENPC1SMN1; SMN2TP53
SCHEMBL20379246 0.87 MMP2 (0.78) RAB9AKDM4ENPC1SMN1; SMN2TP53
SCHEMBL10709034 0.87 MGLL (0.70) RAB9AKDM4ENPC1SMN1; SMN2TP53
SCHEMBL31000016 0.85 MMP2 (0.67) RAB9AKDM4ENPC1SMN1; SMN2TP53
SCHEMBL2247443 0.85 SMN1; SMN2 (1.00) RAB9AKDM4ENPC1SMN1; SMN2TP53
SCHEMBL2245559 0.85 TP53 (0.69) RAB9AKDM4ENPC1SMN1; SMN2TP53
SCHEMBL2248424 0.85 RAB9A (0.78) RAB9AKDM4ENPC1SMN1; SMN2TP53
SCHEMBL27451199 0.84 RAB9A (0.67) RAB9AKDM4ENPC1SMN1; SMN2TP53
SCHEMBL31000021 0.83 MAPT (0.69) RAB9AKDM4ENPC1SMN1; SMN2TP53
SCHEMBL1987139 0.83 MMP2 (1.00) RAB9AKDM4ENPC1SMN1; SMN2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4017873-A2 COMPOSITIONS AND METHODS FOR THE TREATMENT OF PATHOLOGICAL PAIN AND ITCH Duke University (US) 2022-06-29 EP claimed