SCHEMBL29640809

SCHEMBL29640809

O=c1ccnc(-c2ccncn2)n1N1Cc2ccc(F)cc2C1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 14/20 0.36
CYP2D6 P10635 6/20 0.34
CYP1A2 P05177 4/20 0.34
CSNK1A1 P48729 2/20 0.34
GSK3A P49840 1/20 0.34
MAPK9 P45984 2/20 0.33
MAPK10 P53779 1/20 0.33
MAPK11 Q15759 1/20 0.33
MAPK14 Q16539 1/20 0.33
PARP1 P09874 1/20 0.33
PARP10 Q53GL7 1/20 0.33
CDC7 O00311 1/20 0.32
MAP4K4 O95819 1/20 0.32
EGFR P00533 1/20 0.32
FRK P42685 1/20 0.32
DPP4 P27487 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29640865 0.85 GSK3B (0.36) GSK3BCYP2D6CDC7
SCHEMBL29640835 0.70 ADORA2A (0.38) GSK3BCYP2D6CYP1A2CSNK1A1MAPK9
SCHEMBL29640776 0.66 GSK3B (0.37) GSK3BCSNK1A1MAPK9CDC7MAP4K4
SCHEMBL6202952 0.63 GSK3B (0.40) GSK3BCYP2D6CDC7
SCHEMBL29640916 0.60 SMN1; SMN2 (0.41) GSK3BCYP2D6DPP4
SCHEMBL25184191 0.59 MAPK9 (0.47) GSK3BCSNK1A1MAPK9MAPK10MAPK11
SCHEMBL1444770 0.59 KMO (0.51) CYP1A2CSNK1A1MAPK9MAPK10MAPK11
SCHEMBL7482062 0.58 CYP19A1 (0.37) DPP4
SCHEMBL29415406 0.58 MAPK14 (0.57) CYP2D6CSNK1A1MAPK9MAPK10MAPK11
SCHEMBL1445257 0.58 MAPK14 (0.57) CYP2D6CSNK1A1MAPK9MAPK10MAPK11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114502163-A Ethynylheterocycles as RHO-related coiled coil kinase (ROCK) inhibitors 安吉昂生物医药公司 2022-05-13 CN disclosed